TargetAdenosine receptor A1(Mus musculus)
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CCPA from recombinant mouse A1 adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 16.8nMAssay Description:Antagonist activity against adenosine A1 receptor in rat brain membrane in presence of [3H]-R-PIA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 16.8nMAssay Description:Binding affinity to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16.8nMAssay Description:Binding affinity of specific [3H]-R-PIA binding to rat Adenosine A1 receptor in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16.8nMAssay Description:Binding affinity towards rat Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]R-PIA from A1 adenosine receptor in rat brain membranes measured after 3 hrs in presence of adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity against Adenosine A1 receptor labeled by [3H]-CPX in membranes prepared from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Displacement of [125I]IABA from recombinant human A1 adenosine receptor expressed in HEK293 cell membranes measured after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Antagonist activity against human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Antagonist activity against recombinant human adenosine A1 receptor expressed in HEK-293 cells in presence of [125I]-IABA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Binding affinity towards human Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Binding affinity to recombinant human adenosine A1 receptorMore data for this Ligand-Target Pair