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Found 86 with Last Name = 'schuster' and Initial = 'vl'
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85339(17-PHENYL TRINOR PGF2ALPHA-IPR | CAS_130209-76-6 |...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataKi:  23nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85720(AGN 194394)
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM21544((5Z)-7-[(1R,2R,5S)-5-hydroxy-2-[(1E,3S)-3-hydroxyo...)
Affinity DataKi:  38nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM10042((5Z)-7-[(1R,4S,5R,6R)-6-[(1E,3S)-3-hydroxyoct-1-en...)
Affinity DataKi:  38.2nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM21544((5Z)-7-[(1R,2R,5S)-5-hydroxy-2-[(1E,3S)-3-hydroxyo...)
Affinity DataKi:  45nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50020300((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-oct-1-enyl...)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataKi:  45nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50020300((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-oct-1-enyl...)
Affinity DataKi:  48nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85718(AGN 191366)
Affinity DataKi:  71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50390997(CHEMBL1561148)
Affinity DataKi:  71.2nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier organic anion transporter family member 2A1(Mus musculus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM21544((5Z)-7-[(1R,2R,5S)-5-hydroxy-2-[(1E,3S)-3-hydroxyo...)
Affinity DataKi:  98nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Mus musculus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataKi:  104nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50390998(CHEMBL2075005)
Affinity DataKi:  162nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85339(17-PHENYL TRINOR PGF2ALPHA-IPR | CAS_130209-76-6 |...)
Affinity DataKi:  168nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85716(AGN 191995)
Affinity DataKi:  228nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50318491(7-((1R,2S)-2-((S)-3-hydroxyoct-1-enyl)-5-oxocyclop...)
Affinity DataKi:  286nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85715(AGN 191365)
Affinity DataKi:  307nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420244(CHEMBL1628111)
Affinity DataKi:  1.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420245(CHEMBL1614647)
Affinity DataKi:  1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50366524(ESTRONE | ESTROPIPATE | Estrone 3-sulfate | Estron...)
Affinity DataKi:  1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420242(CHEMBL2075012)
Affinity DataKi:  1.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420249(CHEMBL2074598)
Affinity DataKi:  2.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85719(PGF2 Alpha, 1-isopropyl ester)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420251(CHEMBL145704)
Affinity DataKi:  3.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420248(CHEMBL2074651)
Affinity DataKi:  3.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  4.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85719(PGF2 Alpha, 1-isopropyl ester)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50170653((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...)
Affinity DataKi:  5.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataKi:  5.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50390979(BROMOSULFOPHTHALEIN)
Affinity DataKi:  5.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85714(AGN 190911)
Affinity DataKi:  7.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85718(AGN 191366)
Affinity DataKi:  8.13E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420246(CHEMBL2074591)
Affinity DataKi:  9.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50410506(ESTRIOL)
Affinity DataKi:  9.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85714(AGN 190911)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85721(AGN 191088)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85715(AGN 191365)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85717(AGN 192151)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85720(AGN 194394)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85721(AGN 191088)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85716(AGN 191995)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM85717(AGN 192151)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM17639((1S,2S,5R,7S,10R,11S,15S)-5-hydroxy-2,15-dimethylt...)
Affinity DataKi:  1.06E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM17289((1S,10R,11S,15S)-5-hydroxy-15-methyltetracyclo[8.7...)
Affinity DataKi:  1.57E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420250(INDOCYANINE GREEN)
Affinity DataKi:  3.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Rattus norvegicus (Rat))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM25902(4-chloro-2-[(furan-2-ylmethyl)amino]-5-sulfamoylbe...)
Affinity DataKi:  4.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420243(CHEMBL2074705)
Affinity DataKi:  7.62E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1A1(Rattus norvegicus)
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50420247(CHEMBL2074716)
Affinity DataKi: >2.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50366413(PHOSPHOENOLPYRUVATE)
Affinity DataKi:  1.30E+7nMAssay Description:TP_TRANSPORTER: inhibition of PGE2 uptake in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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