Reaction Details Report a problem with these data
Target
Solute carrier organic anion transporter family member 2A1
Ligand
BDBM21544
Substrate
n/a
Meas. Tech.
ChEMBL_836787 (CHEMBL2075312)
Ki
98±n/a nM
Citation
 Pucci, ML; Bao, Y; Chan, B; Itoh, S; Lu, R; Copeland, NG; Gilbert, DJ; Jenkins, NA; Schuster, VL Cloning of mouse prostaglandin transporter PGT cDNA: species-specific substrate affinities. Am J Physiol 277:734-41 (1999) [PubMed]  Article 
Target
Name:
Solute carrier organic anion transporter family member 2A1
Synonyms:
Oatp2a1 | SO2A1_MOUSE | Slc21a2 | Slco2a1 | Solute carrier family 21 member 2
Type:
PROTEIN
Mol. Mass.:
70168.17
Organism:
Mus musculus
Description:
ChEMBL_836787
Residue:
643
Sequence:
MGLLPKPGARQGSGTSSVPARRCSRSVFNNIKVFVLCHGLLQLCQLLYSAYFKSSLTTIEKRFGLSSSSSGLISSLNEISNAILIIFVSYFGSRVNRPRMIGIGGLLLAAGAFVLTLPHFLSEPYQYASTTAGNSSHFQTDLCQKHLPGLLPSKCHSTVPDTQKETSSMWSLMVVAQLLAGVGTVPIQPFGISYVDDFAEPTNSPLYISILFAIAVFGPAFGYLLGSVMLRIFVDYGRVDTATVNLSPGDPRWIGAWWLGLLISSGFLIVTSLPFFFFPRAMSRGAERSVIAEETMKMEEDKSRGSLMDFIKRFPRIFLRLLMNPLFMLVVLSQCTFSSVIAGLSTFLNKFLEKQYDASAAYANLLIGAVNLPAAALGMLFGGILMKRFVFPLQTIPRVAATIMTISIILCAPLFFMGCSTPAVAEVYPPSTPSSIHPQPPACRRDCLCPDSVFHPVCGDNGVEYLSPCHAGCSSLNVSSAASKQPIYLNCSCVTGGSASAKTGSCPTSCAQLLLPSIFLISFVALIACVSHNPLYMMVLRVVNQDEKSFAIGVQFLLMRLLAWLPSPSLYGLLIDSSCIRWNYLCSGRRGACAYYDNDALRNRYLGLQVIYKVLGTLLLFFISWRVKKNREYSLQENASGLI
  
Inhibitor
Name:
BDBM21544
Synonyms:
(5Z)-7-[(1R,2R,5S)-5-hydroxy-2-[(1E,3S)-3-hydroxyoct-1-en-1-yl]-3-oxocyclopentyl]hept-5-enoic acid | 11-Dehydroprostaglandin F2 alpha | Prostaglandin D2 | [3H]PGD2
Type:
radiolabeled ligand
Emp. Form.:
C20H32O5
Mol. Mass.:
352.4651
SMILES:
CCCCC[C@H](O)\C=C\[C@@H]1[C@@H](C\C=C/CCCC(O)=O)[C@@H](O)CC1=O |r|
Structure:
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