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Found 629 with Last Name = 'scipione' and Initial = 'l'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278990(CHEMBL4164524)
Affinity DataKi:  39nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278986(CHEMBL4161860)
Affinity DataKi:  53nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278968(CHEMBL4164186)
Affinity DataKi:  157nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564589(CHEMBL4783436)
Affinity DataKi:  182nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278987(CHEMBL4165299)
Affinity DataKi:  205nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564591(CHEMBL4799735)
Affinity DataKi:  258nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278969(CHEMBL4160790)
Affinity DataKi:  259nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278984(CHEMBL4168710)
Affinity DataKi:  288nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278970(CHEMBL4175914)
Affinity DataKi:  355nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442248(CHEMBL2441983)
Affinity DataKi:  400nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50278983(CHEMBL4172510)
Affinity DataKi:  404nMAssay Description:Mixed inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured from 0.5 to 1.5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442215(CHEMBL2441974)
Affinity DataKi:  450nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564588(CHEMBL4785902)
Affinity DataKi:  450nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442248(CHEMBL2441983)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442215(CHEMBL2441974)
Affinity DataKi:  500nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564584(CHEMBL4791565)
Affinity DataKi:  788nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564585(CHEMBL4780976)
Affinity DataKi:  910nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564592(CHEMBL4798261)
Affinity DataKi:  920nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564590(CHEMBL4778716)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564587(CHEMBL4782376)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564586(CHEMBL4781943)
Affinity DataKi:  1.37E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442209(CHEMBL2441980)
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442209(CHEMBL2441980)
Affinity DataKi:  1.70E+3nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564584(CHEMBL4791565)
Affinity DataKi:  2.36E+3nMAssay Description:Inhibition of equine BChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50564585(CHEMBL4780976)
Affinity DataKi:  2.79E+3nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine as substrate measured for 0.5 to 1.5 mins by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227314(2-(2,6-dichloropyridin-4-ylcarbamoyloxy)-N,N,N-tri...)
Affinity DataKi:  1.95E+4nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227319(2-(dimethylamino)ethyl pyridin-4-ylcarbamate | CHE...)
Affinity DataKi:  2.04E+4nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227314(2-(2,6-dichloropyridin-4-ylcarbamoyloxy)-N,N,N-tri...)
Affinity DataKi:  6.44E+4nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227318(2-(3-bromopyridin-4-ylcarbamoyloxy)-N,N,N-trimethy...)
Affinity DataKi:  1.16E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227315(2-(dimethylamino)ethyl 2,6-dichloropyridin-4-ylcar...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227312(2-(2-chloropyridin-4-ylcarbamoyloxy)-N,N,N-trimeth...)
Affinity DataKi:  1.51E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227313(CHEMBL254299 | N,N,N-trimethyl-2-(pyridin-4-ylcarb...)
Affinity DataKi:  1.59E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227312(2-(2-chloropyridin-4-ylcarbamoyloxy)-N,N,N-trimeth...)
Affinity DataKi:  1.61E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227315(2-(dimethylamino)ethyl 2,6-dichloropyridin-4-ylcar...)
Affinity DataKi:  1.75E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227316(2-(dimethylamino)ethyl 2-chloropyridin-4-ylcarbama...)
Affinity DataKi:  2.08E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227317(2-(dimethylamino)ethyl 3-bromopyridin-4-ylcarbamat...)
Affinity DataKi:  2.73E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227318(2-(3-bromopyridin-4-ylcarbamoyloxy)-N,N,N-trimethy...)
Affinity DataKi:  2.74E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227319(2-(dimethylamino)ethyl pyridin-4-ylcarbamate | CHE...)
Affinity DataKi:  3.14E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227317(2-(dimethylamino)ethyl 3-bromopyridin-4-ylcarbamat...)
Affinity DataKi:  3.16E+5nMAssay Description:Inhibition of acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227316(2-(dimethylamino)ethyl 2-chloropyridin-4-ylcarbama...)
Affinity DataKi:  3.80E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50227313(CHEMBL254299 | N,N,N-trimethyl-2-(pyridin-4-ylcarb...)
Affinity DataKi:  7.54E+5nMAssay Description:Inhibition of butyrylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50466629(CHEMBL4280766)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant HPSE (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  7nMAssay Description:Inhibition of strand transfer activity of recombinant HIV1 integrase using 5'-end-labeled 21-mer double-stranded DNA as substrate after 60 mins by el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  7nMAssay Description:Inhibition of HIV-1 integrase strand transfer activity by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50498306(CHEMBL3582062)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of strand transfer activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human CYP2D6 in presence of NADPH by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human CYP2D6 in presence of NADPH by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50479082(CHEMBL497501)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of strand transfer activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50486615(CHEMBL2236599)
Affinity DataIC50:  15nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of strand transfer activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50498303(CHEMBL3582057)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV-1 integrase assessed as inhibition of strand transfer activity using 32P-labeled DNA as substrate after 1 hr by gel-based assay in ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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