TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH addition measured a...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataKi: 6.00E+4nMAssay Description:Inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human thrombin-mediated platelet aggregation in cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
Affinity DataIC50: 179nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
Affinity DataIC50: 386nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 411nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
Affinity DataIC50: 648nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of (S)-N4-(4-(3-(2-((4-carbamimidoylphenylamino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanamido)butyl)-...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 3.32E+3nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 6.83E+3nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 8.32E+3nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of (S)-N4-(4-(3-(2-((4-carbamimidoylphenylamino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanamido)butyl)-...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.83E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.87E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 3.21E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 3.87E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 5.21E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 6.54E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 6.64E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 7.21E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 7.22E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 7.46E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 7.79E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 8.86E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 8.86E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 9.21E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 9.49E+4nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 9.87E+4nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.79E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.16E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.23E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.45E+5nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.45E+5nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Universidad Nacional De Colombia
Curated by ChEMBL
Universidad Nacional De Colombia
Curated by ChEMBL
Affinity DataIC50: 2.46E+5nMAssay Description:Inhibition of ovine COX-2 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair