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Found 31 with Last Name = 'shaikh' and Initial = 'ms'
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  40nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153386(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-chlorop...)
Affinity DataIC50:  1.80E+3nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50522860(CHEMBL4445442)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis InhA using DDCoA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM13066(2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid...)
Affinity DataIC50:  6.25E+3nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153388(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  8.00E+3nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014170(CHEMBL3260869)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014168(CHEMBL3260867)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014167(CHEMBL3260864)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014166(CHEMBL3260863)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014169(CHEMBL3260868)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153385(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-nitroph...)
Affinity DataIC50:  1.37E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014165(CHEMBL3260862)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM13066(2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014163(CHEMBL3260860)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014162(CHEMBL3260859)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of ovine COX2 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153387(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  1.92E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153387(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  2.38E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153386(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-chlorop...)
Affinity DataIC50:  2.90E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153385(2-(4,5-Dibromo-1H-pyrrole-2-carbonyl)-N-(4-nitroph...)
Affinity DataIC50:  4.21E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153388(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl)-N-(...)
Affinity DataIC50:  4.31E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014170(CHEMBL3260869)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014169(CHEMBL3260868)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014168(CHEMBL3260867)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014167(CHEMBL3260864)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014166(CHEMBL3260863)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014162(CHEMBL3260859)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014163(CHEMBL3260860)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
K.L.E.U'S College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50014165(CHEMBL3260862)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 peroxidase activity assessed as reduction of PGG2 to PGH2 by measuring oxidized TMPD level by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153389(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl-N-(f...)
Affinity DataIC50:  6.03E+4nMpH: 8.5 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-2 in 96-well microtiter plates using succinylated gelatin as the sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Kwazulu-Nata

LigandPNGBDBM153389(2-(1-Methyl-4,5-dibromo-1H-pyrrole-2-carbonyl-N-(f...)
Affinity DataIC50:  8.42E+4nMpH: 8.0 T: 2°CAssay Description:The synthesized compounds were assayed for the inhibitory activities against MMP-12 in 96-well microtiter plates using thiopeptolide as the substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed