Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cerebral membrane after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Displacement of [125I]O-iodo-trans-decalinvesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 13.6nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 60 mins by liquid scintillation counting in presence of DT...More data for this Ligand-Target Pair
Affinity DataKi: 13.8nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 60 mins by liquid scintillation counting in presence of DT...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 15.6nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 20.5nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 60 mins by liquid scintillation counting in presence of DT...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 22.1nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cerebral membrane after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 22.6nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 28.6nMAssay Description:Displacement of [125I]O-iodo-trans-decalinvesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 32.9nMAssay Description:Displacement of [125I]O-iodo-trans-decalinvesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 33.9nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 60 mins by liquid scintillation counting in presence of DT...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 38.3nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 72.5nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-40) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 74.1nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cerebral membrane after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 77.2nMAssay Description:Displacement of [125I]6-iodo-4'-dimethyaminofl avone from beta amyloid (1-42) protein aggregatesMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cerebral membrane after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair