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Found 22 with Last Name = 'shiiki' and Initial = 't'
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322036(CHEMBL1173125 | Ethyl(2S,6S)-4-{[(7-carbamoyl-8H-i...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322037(CHEMBL1173126 | Ethyl(2S,6S)-2,6-dimethyl-4-({[7-(...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322039(CHEMBL1173572 | Ethyl(2S,6S)-2,6-dimethyl-4-{[(7-m...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322043((2S,2'S)-diethyl 2,2'-((5-(2-amino-5-isobutylthiaz...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322041(CHEMBL1172935 | Isopropyl(2S,6S)-4-{[(6,7-dimethyl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317151((2S,2'S)-diethyl 2,2'-(((6,7-dimethyl-8H-indeno[1,...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322042(CHEMBL1172936 | Ethyl4-{[(6,7-dimethyl-8H-indeno[1...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322038(CHEMBL1173571 | Ethyl(2S,6S)-4-[({7-[(2,2-dimethyl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-1,6-bisphosphatase 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50322040(CHEMBL1173636 | Ethyl(2S,6S)-4-{[(7-ethyl-8H-inden...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317154(4-[4-(3-Methoxy-phenyl)-2-oxo-2lambda*5*-[1,3,2]di...)
Affinity DataIC50:  270nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317154(4-[4-(3-Methoxy-phenyl)-2-oxo-2lambda*5*-[1,3,2]di...)
Affinity DataIC50:  300nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317152((2R,4S)-4-[4-(3-Chloro-phenyl)-2-oxo-2lambda*5*-[1...)
Affinity DataIC50:  420nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317151((2S,2'S)-diethyl 2,2'-(((6,7-dimethyl-8H-indeno[1,...)
Affinity DataIC50:  580nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317153(4-[4-(4-Chloro-phenyl)-2-oxo-2lambda*5*-[1,3,2]dio...)
Affinity DataIC50:  650nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317153(4-[4-(4-Chloro-phenyl)-2-oxo-2lambda*5*-[1,3,2]dio...)
Affinity DataIC50:  730nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317157(6,7-Dimethyl-4-(2-oxo-4-pyridin-4-yl-2lambda*5*-[1...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317152((2R,4S)-4-[4-(3-Chloro-phenyl)-2-oxo-2lambda*5*-[1...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317156(6,7-Dimethyl-4-(2-oxo-4-pyridin-3-yl-2lambda*5*-[1...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317159(6,7-Dimethyl-4-[4-(6-methyl-pyridin-3-yl)-2-oxo-2l...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317158(6,7-Dimethyl-4-[4-(2-methyl-pyridin-3-yl)-2-oxo-2l...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317155(6,7-Dimethyl-4-(2-oxo-4-pyridin-2-yl-2lambda*5*-[1...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317160((2R,4S)-6,7-Dimethyl-4-[4-(2-methyl-pyridin-3-yl)-...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed