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Found 183 with Last Name = 'shimazawa' and Initial = 'r'
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145539((2S,4R)-2,4-Dihydroxy-6-[2-[(R)-1-((R)-5-hydroxy-1...)
Affinity DataIC50:  0.5nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066441(2-(2,6-Dimethyl-phenyl)-isoindole-1,3-dione | 2-(2...)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50088679(2-Phenyl-isoindole-1,3-dione | 2-phenyl-1H-isoindo...)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50088679(2-Phenyl-isoindole-1,3-dione | 2-phenyl-1H-isoindo...)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50219329(CHEMBL8968)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066441(2-(2,6-Dimethyl-phenyl)-isoindole-1,3-dione | 2-(2...)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50219329(CHEMBL8968)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity (RA1) against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145538((S)-1-Benzyl-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-dihyd...)
Affinity DataIC50:  1.90nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111216(5-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50: <10nMAssay Description:Inhibitory activity (RA2) against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145540((S)-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-Dihydroxy-2-me...)
Affinity DataIC50:  10nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404242(CHEMBL2114211)
Affinity DataIC50:  30nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404243(CHEMBL2114212 | CHEMBL3350688)
Affinity DataIC50:  50nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50223417(CHEMBL3350292)
Affinity DataIC50: >100nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111221(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-4-nitro-...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111216(5-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111222(4-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111209(2-(2,3,5,6-Tetramethyl-phenyl)-isoindole-1,3-dione...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111217(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-isoindol...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111213(2-(2,3,5-Trimethyl-phenyl)-isoindole-1,3-dione | C...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50070114((+/-)-thalidomide | 2-(2,6-Dioxo-piperidin-3-yl)-i...)
Affinity DataIC50:  370nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111221(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-4-nitro-...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111220(2-(2,4-Dioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl)-is...)
Affinity DataIC50:  440nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147586((S)-4-{2-[(3R,7S)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  440nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  480nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50070114((+/-)-thalidomide | 2-(2,6-Dioxo-piperidin-3-yl)-i...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111211(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-5-nitro-...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111207(2-(2,4-Dioxo-tetrahydro-pyrimidin-1-yl)-isoindole-...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111214(2-[2-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-eth...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111209(2-(2,3,5,6-Tetramethyl-phenyl)-isoindole-1,3-dione...)
Affinity DataIC50:  670nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111217(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-isoindol...)
Affinity DataIC50:  730nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111219(2-(2-Oxo-piperidin-3-yl)-isoindole-1,3-dione | CHE...)
Affinity DataIC50:  850nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  860nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147583((S)-4-Methylene-3-{2-[(R)-7a-(R)-methyl-1-((R)-5-m...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activity; Value ranges from 0.44 uM to 0.89 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111207(2-(2,4-Dioxo-tetrahydro-pyrimidin-1-yl)-isoindole-...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150613(CHEMBL179992 | CHEMBL182645 | [(1R,4S,7aR)-1-(1,5-...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration againsts dual-specificity phosphatase Cell division cycle (Cdc) 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111213(2-(2,3,5-Trimethyl-phenyl)-isoindole-1,3-dione | C...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150612(CHEMBL181402 | CHEMBL182548 | Phosphoric acid mono...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111219(2-(2-Oxo-piperidin-3-yl)-isoindole-1,3-dione | CHE...)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111214(2-[2-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-eth...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibitory activity (RA1) of the compound against Prostaglandin G/H synthase 1 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.44E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111211(2-((R)-3-Methyl-2,6-dioxo-piperidin-3-yl)-5-nitro-...)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261103((Z)-2-(1-hexadecyl-2-oxoindolin-3-ylidene)acetic a...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.62E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50261059((Z)-2-(2-oxo-1-tetradecylindolin-3-ylidene)acetic ...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human Cdc25A phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50150608(2-[1-(1,5-dimethylhexyl)-4,7a-dimethylperhydro-4-i...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration agaunst dual-specificity phosphatase Cell division cycle (Cdc) 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111222(4-Amino-2-((R)-3-methyl-2,6-dioxo-piperidin-3-yl)-...)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibitory activity (RA2) of the compound against Prostaglandin G/H synthase 2 was calculated relative to aspirinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  1.88E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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