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Found 43 with Last Name = 'sisinni' and Initial = 'l'
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataIC50:  21nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human HSP90alpha expressed in Escherichia coli by fluorescence anisotropy methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50126143(Epacadostat | INCB-024360)
Affinity DataIC50:  72nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50126143(Epacadostat | INCB-024360)
Affinity DataIC50:  72nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50031735(CHEMBL3360305)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50361703(CHEMBL1941052)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274536(CHEMBL3900791)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50030791(CHEMBL3342402)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274534(CHEMBL4128056)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50030791(CHEMBL3342402)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274533(CHEMBL4129436)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558530(CHEMBL4749159)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274525(CHEMBL4127843)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558522(CHEMBL4790386)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558539(CHEMBL4744327)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558546(CHEMBL374404)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50361701(CHEMBL1941050)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558528(CHEMBL229510)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558540(CHEMBL4782372)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558538(CHEMBL4800450)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558534(CHEMBL4759143)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558526(CHEMBL4760664)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274518(CHEMBL4128206)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558535(CHEMBL4757189)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558527(CHEMBL389506)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558529(CHEMBL4754880)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558533(CHEMBL4791547)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558531(CHEMBL4747897)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558525(CHEMBL4776062)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558543(CHEMBL4777683)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558521(CHEMBL4755246)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558537(CHEMBL4747344)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50126142(4-Phenylimidazole | CHEMBL14145 | US11053207, Comp...)
Affinity DataIC50:  1.43E+5nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558532(CHEMBL4760024)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558541(CHEMBL372987)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558536(CHEMBL4750312)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558544(CHEMBL4779140)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558545(CHEMBL4741025)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558523(CHEMBL4779268)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558524(CHEMBL4780282)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Alchemical Dynamics

Curated by ChEMBL
LigandPNGBDBM50558542(CHEMBL4779956)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human IDO1 incubated for 60 mins in presence of L-tryptophan by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataKd:  1.5nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human HSP90alpha expressed in Escherichia coli by fluorescence anisotropy methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50274535(CHEMBL4126250)
Affinity DataKd:  10nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) expressed in Escherichia coli BL21-Cod...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed