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Found 280 with Last Name = 'sitaram' and Initial = 'na'
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496157(CHEMBL3121772)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496541(CHEMBL3126811)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496545(CHEMBL3126804)
Affinity DataKi:  2nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496546(CHEMBL3126813)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037243(CHEMBL3356263)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496541(CHEMBL3126811)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037239(CHEMBL3352855)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037237(CHEMBL3356265)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM91678(Pyrazolyl benzenesulfonamide derivative, 7a)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037238(CHEMBL3356264)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496143(CHEMBL3121770)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496533(CHEMBL3126821)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037235(CHEMBL3356266)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human carbonic anhydrase 9 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496154(CHEMBL3121758)
Affinity DataKi:  3nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM91679(Pyrazolyl benzenesulfonamide derivative, 7b)
Affinity DataKi:  3.10nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496158(CHEMBL3121771)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496154(CHEMBL3121758)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037244(CHEMBL3356262)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496149(CHEMBL3121755)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496544(CHEMBL3126807)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human carbonic anhydrase 1-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496546(CHEMBL3126813)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496541(CHEMBL3126811)
Affinity DataKi:  4nMAssay Description:Inhibition of human carbonic anhydrase 2-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM91679(Pyrazolyl benzenesulfonamide derivative, 7b)
Affinity DataKi:  4.20nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM91678(Pyrazolyl benzenesulfonamide derivative, 7a)
Affinity DataKi:  4.30nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496528(CHEMBL3126825)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human carbonic anhydrase 2-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496538(CHEMBL3126820)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496151(CHEMBL3121752)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496528(CHEMBL3126825)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496159(CHEMBL3121769)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496143(CHEMBL3121770)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496156(CHEMBL3121754)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496547(CHEMBL3126824)
Affinity DataKi:  5nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496538(CHEMBL3126820)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496528(CHEMBL3126825)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496535(CHEMBL3126808)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037235(CHEMBL3356266)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human carbonic anhydrase 12 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496154(CHEMBL3121758)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM91679(Pyrazolyl benzenesulfonamide derivative, 7b)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human carbonic anhydrase 2-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496158(CHEMBL3121771)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 12 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase 12 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496530(CHEMBL3126823)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496149(CHEMBL3121755)
Affinity DataKi:  6.5nMAssay Description:Inhibition of human transmembrane carbonic anhydrase 9 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50037231(CHEMBL3356268)
Affinity DataKi:  6.60nMAssay Description:Inhibition of human carbonic anhydrase 12 by stopped flow CO2 hydrase assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496143(CHEMBL3121770)
Affinity DataKi:  6.60nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496157(CHEMBL3121772)
Affinity DataKi:  6.70nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496537(CHEMBL3126805)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496532(CHEMBL3126806)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human carbonic anhydrase 1-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50496547(CHEMBL3126824)
Affinity DataKi:  7.10nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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