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Found 364 with Last Name = 'skalitzky' and Initial = 'd'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145214(2-(4-((methylamino)methyl)phenyl)-1H-benzo[d]imida...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122777(1-Phenyl-8,9-dihydro-7H-2,7,9a-triaza-benzo[cd]azu...)
Affinity DataKi:  4.10nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122775(1-(4-Hydroxymethyl-phenyl)-8,9-dihydro-7H-2,7,9a-t...)
Affinity DataKi:  4.20nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145216(2-(4-{[Bis-(2-hydroxy-ethyl)-amino]-methyl}-phenyl...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145224(2-(4-Dimethylaminomethyl-phenyl)-1H-benzoimidazole...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122781(1-Naphthalen-1-yl-8,9-dihydro-7H-2,7,9a-triaza-ben...)
Affinity DataKi:  4.90nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145223(2-(3-Dimethylaminomethyl-phenyl)-1H-benzoimidazole...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122779(1-(4-Chloro-phenyl)-8,9-dihydro-7H-2,7,9a-triaza-b...)
Affinity DataKi:  5.70nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122776(1-(4-Dimethylaminomethyl-phenyl)-8,9-dihydro-7H-2,...)
Affinity DataKi:  5.80nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145225(2-(4-Pyrrolidin-1-ylmethyl-phenyl)-1H-benzoimidazo...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145221(2-{4-[(4-Methoxy-benzyl)-methyl-amino]-phenyl}-1H-...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194976((S)-2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  6nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122772(1-(3-Dimethylaminomethyl-phenyl)-8,9-dihydro-7H-2,...)
Affinity DataKi:  6.30nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194957(2-((6-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  7nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145219(2-(4-Piperidin-1-ylmethyl-phenyl)-1H-benzoimidazol...)
Affinity DataKi:  7.20nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122774(1-(2-Chloro-phenyl)-8,9-dihydro-7H-2,7,9a-triaza-b...)
Affinity DataKi:  7.70nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145215(2-[4-(4-Methyl-piperazin-1-ylmethyl)-phenyl]-1H-be...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122780(1-(3-Hydroxymethyl-phenyl)-8,9-dihydro-7H-2,7,9a-t...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145222(2-[3-(4-Methyl-piperazin-1-ylmethyl)-phenyl]-1H-be...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145220(2-(3-Pyrrolidin-1-ylmethyl-phenyl)-1H-benzoimidazo...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194955(2-((6-(2-(2-(3-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  11nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122773(1-(3-Trifluoromethyl-phenyl)-8,9-dihydro-7H-2,7,9a...)
Affinity DataKi:  11.2nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145217(2-(4-Morpholin-4-ylmethyl-phenyl)-1H-benzoimidazol...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145218(2-(3-Piperidin-1-ylmethyl-phenyl)-1H-benzoimidazol...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM27091(2-phenyl-1H-1,3-benzodiazole-4-carboxamide | CHEMB...)
Affinity DataKi:  15nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194971(2-((6-(2-(5-methyl-2-(3-(trifluoromethyl)phenyl)ox...)
Affinity DataKi:  15nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194968(3-(6-(4-(3-chlorophenoxy)-2-methylphenethoxy)pyrid...)
Affinity DataKi:  15nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194961(2-((6-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  16nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194950(2-((6-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  17nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194974(2-((6-(2-(5-methyl-2-p-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  23nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145212(2-(3-Morpholin-4-ylmethyl-phenyl)-1H-benzoimidazol...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194967(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  38nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50122778(1-Methyl-8,9-dihydro-7H-2,7,9a-triaza-benzo[cd]azu...)
Affinity DataKi:  45nMAssay Description:Inhibitory activity of the compound against human full length Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194969(2-((6-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  52nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194963(2-methoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataKi:  63nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194952(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  81nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194970(2-((6-(2-(5-methyl-2-(4-(trifluoromethyl)phenyl)ox...)
Affinity DataKi:  94nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194953(2-ethoxy-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataKi:  150nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194977(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  240nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194965((S)-2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenylo...)
Affinity DataKi:  270nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50145213(2-(3-{[Bis-(2-hydroxy-ethyl)-amino]-methyl}-phenyl...)
Affinity DataKi:  272nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataKi:  334nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194956(4-methyl-2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataKi:  360nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194960(1-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  394nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  440nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194975(2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazo...)
Affinity DataKi:  560nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194958(2-((6-(3-(5-methyl-2-phenyloxazol-4-yl)propoxy)pyr...)
Affinity DataKi:  810nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194954(2-((6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50194951(2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM27506(3-AB | 3-aminobenzamide | CHEMBL81977)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity towards human poly(ADP-ribose) polymerase-1 (PARP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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