Affinity DataKi: 0.990nMAssay Description:Binding affinity to NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at human NR1a/NR2B receptor expressed in mouse fibroblast LMTK cells assessed as inhibition of Glu/Gly induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-Ro-256981 from recombinant NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity against NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-Ro-256981 from recombinant NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]-Ro-256981 from recombinant NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]-Ro-256981 from recombinant NR1/NR2B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at NR1/NR2B receptor assessed as inhibition of Glu/Gly induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human NR1a/NR2B receptor expressed in mouse fibroblast LMTK cells assessed as inhibition of Glu/Gly induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Antagonist activity at NR1/NR2B receptor assessed as inhibition of Glu/Gly induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 177nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 209nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Antagonist activity against NR1/NR2B receptor expressed in xenopus oocytes assessed as inhibition of NMDA induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Antagonist activity against NR1a/NR2B receptor transfected in human HEK293 cells assessed as inhibition of NMDA-induced Ca2+ influxMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 5.10nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain straitumMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 15.2nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain thalamusMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 5.40nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain thalamusMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 5.90nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain olfactory tubercleMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 1.90nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain olfactory tubercleMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 9.30nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain straitumMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 9.80nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain cortexMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 3.20nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain cortexMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 7.10nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain hippocampusMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Institute Of Biomedical Imaging (I2Bm)
Curated by ChEMBL
Affinity DataKd: 9.10nMAssay Description:Binding affinity to NMDAR NR2B in Sprague-Dawley rat brain hippocampusMore data for this Ligand-Target Pair