Affinity DataKi: 0.0470nMAssay Description:Compound was evaluated for the inhibition of human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nM ΔG°: -51.7kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity against serine protease factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity (in vitro) of the compound towards human Coagulation factor X was determined at 10 mg/kg peroral doseMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nM ΔG°: -51.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nM ΔG°: -51.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nM ΔG°: -50.6kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity (in vitro) of the compound towards human Coagulation factor X was determined at 5 mg/kg peroral doseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Compound was evaluated for the inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nM ΔG°: -50.2kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against serine protease factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DPDPE from human DOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory activity against human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against serine protease Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against serine protease factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against serine protease factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against serine protease factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity (in vitro) of the compound towards human Coagulation factor X was determined at 10 mg/kg peroral doseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inibition of Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against serine protease Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.5kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair