Affinity DataKi: 0.200nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from rat brain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from rat brain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from rat brain membrane using [3H]DAMGOMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Combichem
Curated by ChEMBL
Combichem
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Evaluated for binding affinity against alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Compound was evaluated for binding affinity towards mu-specific opiate receptor from combinatorial peptoid libraryMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:The inhibitory constant of the compound was evaluated against Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:The inhibitory constant of the compound was evaluated against Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:The inhibitory constant of the compound was evaluated against Endothelin A receptor in rabbit renal artery tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:The compound was tested for the binding affinity against eEndothelin A receptor in murine 3T3 cells using [125I]-ET-1 as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:The inhibitory constant of the compound was evaluated against Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <800nMAssay Description:The inhibitory constant was evaluated against Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cellsMore data for this Ligand-Target Pair