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Found 30 with Last Name = 'sperotto' and Initial = 'n'
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531739(MA-1 | TPI (freebase) | Tipiracil)
Affinity DataKi:  20nMAssay Description:Competitive inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531739(MA-1 | TPI (freebase) | Tipiracil)
Affinity DataIC50:  35nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50122770(6-Amino-5-bromo-1H-pyrimidine-2,4-dione | 6-Amino-...)
Affinity DataIC50:  35nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531729(CHEMBL4469338)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531734(CHEMBL4468378)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531742(CHEMBL4579188)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531736(CHEMBL4438928)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531740(CHEMBL4445259)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531737(CHEMBL4527207)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-(+)-mephenytoin as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2E1(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2E1 in human liver microsomes using chlorzoxazone as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using tolbutamide as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50234734(CHEMBL4094462)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate by HPLC-MS/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531738(CHEMBL4542724)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531735(CHEMBL4435521)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531731(CHEMBL4439474)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531743(CHEMBL4472112)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50134399(1,7-Dihydro-pyrrolo[2,3-d]pyrimidine-2,4-dione | 7...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531741(CHEMBL4579033)
Affinity DataIC50:  8.70E+4nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP3A4 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531730(CHEMBL4582134)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2C19 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2E1(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2E1 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Universidade Federal Do Pampa

Curated by ChEMBL
LigandPNGBDBM50531733(CHEMBL4464628)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human thymidine phosphorylase expressed in Escherichia coli Rosetta (DE3) cells using thymidine as substrate after 1 min by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Pontif£Cia Universidade Cat£Lica Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50531732(CHEMBL4455140)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2C9 in human liver microsomes by HPLC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed