Affinity DataKi: 0.420nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human plasma carboxypeptidase NMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of bovine pancreatic carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 111nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of VMAT2 in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 206nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 269nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 278nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 344nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: >700nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [3H]-25-hydroxycholesterol from His-Flag-tagged human RORgammat LBD (309 to 508 residues) expressed in Escherichia coli measured afte...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma carboxypeptidase NMore data for this Ligand-Target Pair
Affinity DataKi: >1.55E+4nMAssay Description:Binding affinity to RORalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Inhibition of human TAFIaMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to RORbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0200nMAssay Description:Transrepression of glucocorticoid receptor in human PBMC assessed as inhibition of LPS induced TNF alpha release preincubated for 45 mins followed by...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0290nMAssay Description:Transrepression of glucocorticoid receptor in PMA-stimulated human ChaGoK1 cells expressing TRE-LacZ construct assessed as inhibition of AP-1 mediate...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0320nMAssay Description:Transrepression of glucocorticoid receptor in PMA-stimulated human ChaGoK1 cells expressing TRE-LacZ construct assessed as inhibition of AP-1 mediate...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0370nMAssay Description:Displacement of fluormone labelled GS Red from human recombinant glucocorticoid receptor after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Transrepression of glucocorticoid receptor in PMA-stimulated human ChaGoK1 cells expressing TRE-LacZ construct assessed as inhibition of AP-1 mediate...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0440nMAssay Description:Displacement of fluormone labelled GS Red from human recombinant glucocorticoid receptor after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0490nMAssay Description:Transrepression of glucocorticoid receptor in PMA-stimulated human ChaGoK1 cells expressing TRE-LacZ construct assessed as inhibition of AP-1 mediate...More data for this Ligand-Target Pair