Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-alpha' and Ligand = 'BDBM302860'
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM302860((2S)-1-(3-Thienyl)propan-2-ol | US9598431, 3)
Affinity DataKi: >1.55E+4nMAssay Description:Binding affinity to RORalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Lilly Research Laboratories

Curated by ChEMBL
LigandPNGBDBM302860((2S)-1-(3-Thienyl)propan-2-ol | US9598431, 3)
Affinity DataKi: >2.04E+4nMAssay Description:Receptor competition binding assays are run in a buffer made up of DPBS (1 L) (Hyclone #SH30028.03), 2.2 g BSA Fraction v (Roche #9048-46-8), 100 mL ...More data for this Ligand-Target Pair
In DepthDetails US Patent