Compile Data Set for Download or QSAR
maximum 50k data
Found 72 with Last Name = 'strehle' and Initial = 'a'
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273003(CHEMBL456781 | [5-(2-Amino-ethyl)-3H-[1,3,4]oxadia...)
Affinity DataIC50:  7.40E+3nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273043(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-thione Hydroch...)
Affinity DataIC50:  4.90E+4nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273004(5-Piperidin-4-yl-3H-[1,3,4]oxadiazol-2-thione Hydr...)
Affinity DataIC50:  5.90E+4nMAssay Description:Agonist activity at rat wild type GABAAalpha1beta2 receptor expressed in Xenopus laevis oocytes as inhibition of GABA-induced current at -60 mV by Tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273004(5-Piperidin-4-yl-3H-[1,3,4]oxadiazol-2-thione Hydr...)
Affinity DataIC50:  6.60E+4nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273110(4-(5-Methyl-[1,3,4]oxadiazol-2-yl)-piperidine Hydr...)
Affinity DataIC50:  7.60E+4nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273001(5-Piperidin-4-yl-3H-[1,3,4]oxadiazol-2-one Hydroch...)
Affinity DataIC50:  1.23E+5nMAssay Description:Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50050950(Betulinic acid | CHEMBL37 | Dihydrobetulinic acid)
Affinity DataEC50:  2.17E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273004(5-Piperidin-4-yl-3H-[1,3,4]oxadiazol-2-thione Hydr...)
Affinity DataEC50:  9.50E+6nMAssay Description:Agonist activity at rat wild type GABAAalpha1beta2 receptor expressed in Xenopus laevis oocytes at -60 mV by Two-Electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataEC50:  1.00E+4nMAssay Description:Activity at rat wild type GABAAalpha1beta2 receptor expressed in Xenopus laevis oocytes at -60 mV by Two-Electrode voltage clamp methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  2.80E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha1beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  1.82E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha2beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  2.30E+6nMAssay Description:Agonist activity at rat recombinant GABAAalpha3beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  1.28E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha4beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  1.37E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha5beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-6(RAT)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at rat recombinant GABAAalpha6beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50236238((3alpha,5beta)-3-hydroxycholan-24-oic acid | 3alph...)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataEC50:  1.04E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50346601(NSC-114945 | OLEANOLIC_ACID | Oleanolic acid | Ole...)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303455((5beta,8alpha,14beta,18beta,19beta)-3-[(Isobutyryl...)
Affinity DataEC50:  3.65E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303456(3-Methoxylupan-28-oic Acid | CHEMBL567770)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303457(Benzyl 3-Hydroxylup-20(29)-en-28-oate | CHEMBL5715...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303458(Benzyl 3-Methoxylup-20(29)-en-28-oate | CHEMBL5771...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303459((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13aR,13bR)-9-ally...)
Affinity DataEC50:  2.08E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303460((1R,3aS,5aR,5bR,7aR,9R,11aR,11bR,13aR,13bR)-9-ally...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303461((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13bR)-9-hydroxy-5...)
Affinity DataEC50:  6.27E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303462((1R,3aS,5aR,5bR,7aR,9R,11aR,11bR,13bR)-9-hydroxy-5...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303463(20(R)-20(29)-Epoxybetulinic Acid | 9-Hydroxy-5alph...)
Affinity DataEC50:  6.91E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303464(29-Dihydroxylupan-28-oic Acid | CHEMBL583203)
Affinity DataEC50:  3.32E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50103962((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13aR,13bS)-1-Acet...)
Affinity DataEC50:  3.11E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303465(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethyl 3-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303466(2-[(tert-butoxycarbonyl)amino]ethyl 3-hydroxylup-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303467(CHEMBL576519 | Pyridin-4-ylmethyl 3-hydroxylup-20(...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303468(({[3-hydroxy-28-oxolup-20(29)-en-28-yl]oxy}methyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303469(CHEMBL583640 | N-cyclopropyl-3-hydroxylup-20(29)-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303470(3-hydroxylup-20(29)-en-28-amide | CHEMBL583224)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303471((1R,3alphaS,5alphaR,5betaR,9S,11aR)-N-(carbamoylme...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303472(3-hydroxy-N-[2-(2-hydroxyethoxy)ethyl]lup-20(29)-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303473(3-hydroxy-N-[4-hydroxy-2-(hydroxymethyl)butyl]lup-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303474(CHEMBL571516 | N-(2,3-dihydroxypropyl)-3-hydroxylu...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303475(3-hydroxy-N-(2-hydroxyethyl)lup-20(29)-en-28-amide...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303476(3-hydroxy-N-(4-hydroxybutyl)lup-20(29)-en-28-amide...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303477(CHEMBL576716 | Ethyl N-[3-hydroxy-28-oxolup-20(29)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303478(CHEMBL429204 | N-[3-hydroxy-28-oxolup-20(29)-en-28...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50240501((1R,3aS,5aR,5bR,7aR,9S,11aR,11bR,13aR)-methyl 9-hy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303479(3alpha-isocyanato-1-isopropenyl-5alpha,5beta,8,8,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303480(CHEMBL576520 | N-cyclopropyl-N'-(9-hydroxy-1-isopr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303481(CHEMBL571736 | N-(2-hydroxyethyl)-N'-(9-hydroxy-1-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50303482(1-((1R,3alphaS,5alphaR,5betaR,9S,11alphaR)-icosahy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 72 total ) | Next | Last >>
Jump to: