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Found 966 with Last Name = 'suga' and Initial = 'h'
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM223314(YPYSCWARHVRIREN | piHA-D1)
Affinity DataKi:  1nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239342(CHEMBL4075127)
Affinity DataKi:  1nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50052910(CHEMBL118271 | N-[4-(5-Hydroxy-2,3,4,5-tetrahydro-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239349(CHEMBL4104877)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239344(CHEMBL4094707)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM223315(YPYSCWVRHSDPHKF | piHA-D3)
Affinity DataKi:  2.70nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239346(CHEMBL4064556)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239347(CHEMBL4086079)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239349(CHEMBL4104877)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239348(CHEMBL4102459)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239343(CHEMBL4076436)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM223316(YPYSCWVRH | piHA-Dm)
Affinity DataKi:  7nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50052910(CHEMBL118271 | N-[4-(5-Hydroxy-2,3,4,5-tetrahydro-...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239342(CHEMBL4075127)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079268(CHEMBL3416766)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239344(CHEMBL4094707)
Affinity DataKi:  46nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079261(CHEMBL3416768)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239347(CHEMBL4086079)
Affinity DataKi:  54nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079268(CHEMBL3416766)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239345(CHEMBL4078185)
Affinity DataKi:  78nMAssay Description:Displacement of [125I] phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 from human recombinant vasopressin V1a receptor expressed in HEK293 aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079266(CHEMBL3416774)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239346(CHEMBL4064556)
Affinity DataKi:  140nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239343(CHEMBL4076436)
Affinity DataKi:  160nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239348(CHEMBL4102459)
Affinity DataKi:  170nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079269(CHEMBL3416767)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508772(CHEMBL4452943)
Affinity DataKi:  440nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079263(CHEMBL3416770)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079265(CHEMBL3416773)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508769(CHEMBL4483351)
Affinity DataKi:  800nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079263(CHEMBL3416770)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079263(CHEMBL3416770)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079264(CHEMBL3416772)
Affinity DataKi:  870nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079262(CHEMBL3416769)
Affinity DataKi:  870nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079261(CHEMBL3416768)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50079262(CHEMBL3416769)
Affinity DataKi:  910nMAssay Description:Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50239345(CHEMBL4078185)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [3H] (Arg8)-vasopressin from human vasopressin V2 receptor expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508771(CHEMBL4555617)
Affinity DataKi:  2.00E+3nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508774(CHEMBL4538618)
Affinity DataKi:  3.50E+3nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508770(CHEMBL4454475)
Affinity DataKi:  2.04E+4nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50508773(CHEMBL4589938)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of C-terminal His6-tagged linked Zika virus NS2B-NS3 protease domain expressed in Escherichia coli Bl21(DE3) using Bz-Nle-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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