TargetBromodomain-containing protein 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma
Curated by ChEMBL
Mitsubishi Tanabe Pharma
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of Flag-tagged BRD4 (unknown origin)-biotinylated AcH4 (Lys5, 8, 12, 16) histone peptide binding expressed in CHO cells after 60 mins by T...More data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to RAP1A in human RBC membrane by western blot analysisMore data for this Ligand-Target Pair
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to RAP1A in human RBC membrane by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to RAP1A in human RBC membrane by surface plasmon resonance analysis with inverted configurationMore data for this Ligand-Target Pair