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Found 59 with Last Name = 'tan' and Initial = 'uk'
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of Aurora B kinaseMore data for this Ligand-Target Pair
TargetAurora kinase C(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of Aurora C kinaseMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  13nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase C(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  61nMAssay Description:Inhibition of Aurora C kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12985(5-Amido-pyrrolopyrazole 9d | CHEMBL402548 | N-{5-[...)
Affinity DataKi:  79nMAssay Description:Inhibition of Aurora B kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479526(CHEMBL515560)
Affinity DataIC50:  33nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479524(CHEMBL474344)
Affinity DataIC50:  449nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479510(CHEMBL515112)
Affinity DataIC50:  460nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479520(CHEMBL473334)
Affinity DataIC50:  719nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479527(CHEMBL461954)
Affinity DataIC50:  804nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479521(CHEMBL461785)
Affinity DataIC50:  838nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479522(CHEMBL473131)
Affinity DataIC50:  960nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479528(CHEMBL518032)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479511(CHEMBL474540)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479517(CHEMBL461599)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479525(CHEMBL473333)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479531(CHEMBL517573)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479512(CHEMBL516353)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479529(CHEMBL514951)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479516(CHEMBL460720)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479519(CHEMBL461784)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479513(CHEMBL460905)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479533(CHEMBL460728)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479518(CHEMBL461972)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479509(CHEMBL473948)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479530(CHEMBL517571)
Affinity DataIC50:  5.25E+3nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50372019(CHEMBL402349)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50372021(CHEMBL271894)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479514(CHEMBL454390)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479515(CHEMBL455180)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50372017(CHEMBL1589017)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479534(CHEMBL455177)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50372020(CHEMBL439417)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50372018(CHEMBL255808)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479532(CHEMBL451034)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50479523(CHEMBL461955)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Aurora kinase A T288D mutant expressed in Escherichia coli BL21 DE3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  220nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50181911((5-{3-[(6-BENZOYL-1-PROPYL-2-NAPHTHYL)OXY]PROPOXY}...)
Affinity DataEC50:  8nMAssay Description:Activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196245(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196246(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50181911((5-{3-[(6-BENZOYL-1-PROPYL-2-NAPHTHYL)OXY]PROPOXY}...)
Affinity DataEC50:  500nMAssay Description:Activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50181911((5-{3-[(6-BENZOYL-1-PROPYL-2-NAPHTHYL)OXY]PROPOXY}...)
Affinity DataEC50:  70nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196245(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  2.21E+3nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196247(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  2.08E+3nMAssay Description:Activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196246(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  650nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196248(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  1.10E+3nMAssay Description:Activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196249(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196250(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  4.30E+3nMAssay Description:Activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196250(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  210nMAssay Description:Activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
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