Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Tokyo Medical And Dental University (Tmdu)
Curated by ChEMBL
Affinity DataKi: 199nMAssay Description:Displacement of [3H]ketanserin from Sprague-Dawley rat cerebral cortex 5-HT2A receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity against GST-hARLBD was measured in SC-3 cell by using [3H]-testosterone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.38E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Displacement of [3H]testosterone from wild type human androgen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0480nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair