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Found 4 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor' and Ligand = 'BDBM50565950'
TargetVitamin D3 receptor(Bos taurus)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565950(CHEMBL4776651)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565950(CHEMBL4776651)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human VDR expressed in HEK293 cells expressing mouse osteopontin VDRE assessed as induction of receptor transactivation incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565950(CHEMBL4776651)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human VDR expressed in African green monkey COS7 cells expressing mouse osteopontin VDRE assessed as induction of receptor transa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50565950(CHEMBL4776651)
Affinity DataEC50:  0.530nMAssay Description:Agonist activity at VDR in human HL-60 cells assessed as induction of cell differentiation of promyelocytes to monocytes after 4 days by NBT reductio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed