Affinity DataKi: 0.510nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX iradioligand n membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for adenosine A2a receptor by using as [3H]-ZM-241,385 radioligand in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 1.02nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 1.13nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against Adenosine A2b receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for inhibition of calf intestinal mucosa adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for adenosine A1 receptor determined using hamster DDT1 cell membranes with [3H]-CCPA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.74nMAssay Description:Inhibition of Adenosine deaminase (ADA) of calf intestineMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against Adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes prepared from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity against Adenosine A1 receptor labeled by [3H]-CPX in membranes prepared from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity for adenosine A1 receptor determined using hamster DDT1 cell membranes with [3H]-CCPA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]CPX from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 19.5+/-12.0More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair