Affinity DataKi: 43nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Inhibition of N-terminal His-tagged Zika virus NS2B (46 to 99 residues) - NS3 (1 to 187 residues) protease domain expressed in Rosetta2-(DE3) assesse...More data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.05E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.21E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 2.86E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.07E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.13E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.28E+4nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 4.37E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 4.74E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.14E+4nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 8.29E+4nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 1.09E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 1.38E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.78E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 1.93E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of N-terminal His6-tagged Zika virus NS2B (45 to 96 residues) - NS3 (1 to 177 residues) protease domain expressed in Escherichia coli Bl21...More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of N-terminal His-tagged Zika virus NS2B (49 to 95 residues) - NS3 (1 to 185 residues) protease domain expressed in Escherichia coli Bl21(...More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of N-terminal unlinked Zika virus NS2B (45 to 96 residues) - NS3 (1 to 177 residues) protease domain expressed in Escherichia coli Bl21(DE...More data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:Inhibition of N-terminal unlinked Zika virus NS2B (45 to 96 residues) - NS3 (1 to 177 residues) protease domain expressed in Escherichia coli Bl21(DE...More data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Inhibition of N-terminal unlinked Zika virus NS2B (45 to 96 residues) - NS3 (1 to 177 residues) protease domain expressed in Escherichia coli Bl21(DE...More data for this Ligand-Target Pair
TargetGenome polyprotein [1394-1440]/[1476-1660,T1585M](Dengue virus 3 (strain S221/03))
Novartis Institute For Tropical Diseases
Novartis Institute For Tropical Diseases
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitors were assayed in a 96-well plate format. Typically, protease was preincubated with concentrations of test compounds at 37 deg C for 30 min....More data for this Ligand-Target Pair
TargetGenome polyprotein [1066-1250,R1182K]/[1394-1440,K1405R,D1408E](Dengue virus 2 (strain TSV01))
Novartis Institute For Tropical Diseases
Novartis Institute For Tropical Diseases
Affinity DataIC50: 1.10E+3nM Kd: 7.70E+3nMpH: 7.5 T: 2°CAssay Description:Inhibitors were assayed in a 96-well plate format. Typically, protease was preincubated with concentrations of test compounds at 37 deg C for 30 min....More data for this Ligand-Target Pair