Compile Data Set for Download or QSAR
maximum 50k data
Found 28 with Last Name = 'veeneman' and Initial = 'g'
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076948((R)-1-((3R,4R,4aR)-Decahydro-isoquinoline-1-carbon...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076945((S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-prop...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076949((S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-prop...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076952(3-{[(S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076953((R)-1-(3,3-Diphenyl-propionyl)-pyrrolidine-2-carbo...)
Affinity DataIC50:  260nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076951(((R)-2-Cyclohexyl-1-{methyl-[(2-oxo-1-piperidin-4-...)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076946((S)-N-Benzyl-2-oxo-3-[2-(2-oxo-3-phenylmethanesulf...)
Affinity DataIC50:  590nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076954(((R)-2-Cyclohexyl-1-{[(2-oxo-1-piperidin-4-ylmethy...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076947((S)-N-Benzyl-2-oxo-3-[2-(2-oxo-3-phenylmethanesulf...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076945((S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-prop...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076948((R)-1-((3R,4R,4aR)-Decahydro-isoquinoline-1-carbon...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076950(CHEMBL284008 | {(R)-2-Cyclohexyl-1-[(S)-1-(2-oxo-1...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076946((S)-N-Benzyl-2-oxo-3-[2-(2-oxo-3-phenylmethanesulf...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076949((S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-prop...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076951(((R)-2-Cyclohexyl-1-{methyl-[(2-oxo-1-piperidin-4-...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076947((S)-N-Benzyl-2-oxo-3-[2-(2-oxo-3-phenylmethanesulf...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076950(CHEMBL284008 | {(R)-2-Cyclohexyl-1-[(S)-1-(2-oxo-1...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076952(3-{[(S)-1-((R)-3-Cyclohexyl-2-ethanesulfonylamino-...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076954(((R)-2-Cyclohexyl-1-{[(2-oxo-1-piperidin-4-ylmethy...)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibitory activity against thrombin with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50076953((R)-1-(3,3-Diphenyl-propionyl)-pyrrolidine-2-carbo...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibitory activity against Coagulation factor X with respect to ArgatrobanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataIC50:  1.34E+5nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50131559(6-Hydroxy-2-(4-methoxy-phenyl)-3-methyl-chroman-4-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM25862(4-[3-(4-hydroxyphenyl)phenyl]phenol | CHEMBL66279 ...)
Affinity DataEC50:  800nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50131558(4-[3,5-di(4-hydroxyphenyl)phenyl]phenol | CHEMBL11...)
Affinity DataEC50:  80nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50131557(CHEMBL116918 | [1,1';4',1'']Terphenyl-4,4''-diol)
Affinity DataEC50:  1.20E+3nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50131556(6-Hydroxy-2-(4-hydroxy-phenyl)-3-methyl-chroman-4-...)
Affinity DataEC50:  4nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50131560(4,4''-Dimethoxy-[1,1';3',1'']terphenyl | CHEMBL665...)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional agonist activity in Chinese hamster ovary cells expressing human Estrogen Receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed