Compile Data Set for Download or QSAR
maximum 50k data
Found 20 with Last Name = 'venkitaraman' and Initial = 'ar'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM5485(6-(cyclohexylmethoxy)-9H-purin-2-amine | CHEMBL269...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM5594(2-arylamino-pyrimidine deriv. 9d | 4-{[4-amino-6-(...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590137(CHEMBL5198078)
Affinity DataIC50:  5.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590138(CHEMBL5201730)
Affinity DataIC50:  6.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590134(CHEMBL5180335)
Affinity DataIC50:  1.10E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590135(CHEMBL5180822)
Affinity DataIC50:  1.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590136(CHEMBL5203610)
Affinity DataIC50:  1.90E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590133(CHEMBL5184713)
Affinity DataIC50:  8.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590132(CHEMBL5202453)
Affinity DataIC50:  3.33E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50099398(5-Bromo-1H-indazole | CHEMBL16425 | cid_761929)
Affinity DataIC50:  4.10E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590137(CHEMBL5198078)
Affinity DataKd:  1.02E+4nMAssay Description:Binding affinity to CK2alpha (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM50159250(2-Naphthol | 2-naphthalenol | CHEMBL14126 | Naphth...)
Affinity DataKd:  4.60E+5nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM23450(1-Naphthalenol | 1-Naphthol | CHEMBL122617 | Napht...)
Affinity DataKd:  4.30E+5nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM93044(L-Methyl ester tryptophan, 8)
Affinity DataKd:  5.70E+5nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM50335100(1,3-benzothiazol-2-amine | 2-Aminobenzothiazole, 6...)
Affinity DataKd:  7.30E+5nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM24627(1H-indazole | Indazole, 5 | Indazole, 6)
Affinity DataKd:  1.00E+6nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM93043(4-Methylester indole, 4)
Affinity DataKd:  1.30E+6nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590138(CHEMBL5201730)
Affinity DataKd:  1.58E+4nMAssay Description:Binding affinity to CK2alpha (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM32212(1H-indol-5-ol | cid_16054)
Affinity DataKd:  2.10E+6nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair
TargetDNA repair and recombination protein RadA(Pyrococcus furiosus)
University of Cambridge

LigandPNGBDBM93042(Indole, 2)
Affinity DataKd:  2.10E+6nMAssay Description:The thermal-shift denaturation assay was performed on an iCycler iQ Real Time Detection System (BioRad) in 96-well iCycler iQ PCR plates sealed with ...More data for this Ligand-Target Pair