Affinity DataKi: 150nMAssay Description:Binding affinity at iGluR1o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity at iGluR3o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Binding affinity at iGluR4o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:Binding affinity at iGluR1o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Binding affinity at iGluR2o(R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 273nMAssay Description:Binding affinity at iGluR2o(R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 323nMAssay Description:Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 531nMAssay Description:Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+3nMAssay Description:Binding affinity at iGluR4o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity at iGluR3o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at iGluR5(Q) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.85E+4nMAssay Description:Binding affinity at iGluR5(Q) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity at iGluR6(V,C,R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity at iGluR6(V,C,R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0407nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0427nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0447nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0501nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0525nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0603nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0631nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0646nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0741nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0741nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0759nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0794nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0794nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0832nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0871nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0891nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0933nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0977nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.107nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.112nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.115nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.132nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.132nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.151nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.155nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.158nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.166nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.209nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.245nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.245nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.263nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.275nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.288nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.288nMAssay Description:Displacement of [125I]-CCK-8 from human CCK2R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair