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Found 299 with Last Name = 'villalobos' and Initial = 'a'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474703(CHEMBL1269)
Affinity DataKi: <6nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474703(CHEMBL1269)
Affinity DataKi: <6nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474703(CHEMBL1269)
Affinity DataKi: <6nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  6.62nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50185474((+)-4-(3-(4-chlorophenyl)-3-hydroxypyrrolidin-1-yl...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474702(CHEMBL358190)
Affinity DataKi:  6.71nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474706(CHEMBL148626)
Affinity DataKi:  6.72nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474708(CHEMBL149877)
Affinity DataKi:  6.78nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474706(CHEMBL148626)
Affinity DataKi:  6.79nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  6.87nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474705(CHEMBL357956)
Affinity DataKi:  6.91nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474700(CHEMBL149721)
Affinity DataKi:  6.96nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474700(CHEMBL149721)
Affinity DataKi:  7.11nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474705(CHEMBL357956)
Affinity DataKi:  7.11nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474709(CHEMBL147829)
Affinity DataKi:  7.23nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  7.27nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474701(CHEMBL147830)
Affinity DataKi:  7.34nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474708(CHEMBL149877)
Affinity DataKi:  7.36nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50185474((+)-4-(3-(4-chlorophenyl)-3-hydroxypyrrolidin-1-yl...)
Affinity DataKi:  7.48nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474702(CHEMBL358190)
Affinity DataKi:  7.49nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474706(CHEMBL148626)
Affinity DataKi:  7.58nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474701(CHEMBL147830)
Affinity DataKi:  7.59nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474705(CHEMBL357956)
Affinity DataKi:  7.62nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474708(CHEMBL149877)
Affinity DataKi:  7.62nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474702(CHEMBL358190)
Affinity DataKi:  7.64nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474700(CHEMBL149721)
Affinity DataKi:  7.81nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474701(CHEMBL147830)
Affinity DataKi:  7.81nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474707(CHEMBL148627)
Affinity DataKi:  7.81nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474707(CHEMBL148627)
Affinity DataKi:  7.82nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50185474((+)-4-(3-(4-chlorophenyl)-3-hydroxypyrrolidin-1-yl...)
Affinity DataKi:  7.98nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.98nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474707(CHEMBL148627)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474709(CHEMBL147829)
Affinity DataKi:  8.05nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474704(CHEMBL148794)
Affinity DataKi:  8.07nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474704(CHEMBL148794)
Affinity DataKi:  8.09nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474709(CHEMBL147829)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  8.34nMAssay Description:Displacement of [3H]7-OH-DPAT from human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM50474704(CHEMBL148794)
Affinity DataKi:  8.96nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A And M University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  9.05nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM223332(US9315520, 19 | US9605007, Example 19 | US9744173,...)
Affinity DataIC50:  0.0140nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50452875(CHEMBL4212046)
Affinity DataIC50:  0.0330nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50452884(CHEMBL4217023)
Affinity DataIC50:  0.0340nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50452883(CHEMBL4203860)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50032162(3-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-5,7-dihydro-...)
Affinity DataIC50:  0.330nMAssay Description:In vitro inhibition of Acetylcholinesterase from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM47353(BDBM143220 | US9029362, 173 | US9687494, 25)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of human BACE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50032161(3-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-7-methyl-5,7...)
Affinity DataIC50:  0.480nMAssay Description:In vitro inhibition of Acetylcholinesterase from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM143218(US8940748, 34 | US9029362, 34 | US9687494, 34)
Affinity DataIC50: <0.540nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50032164(3-(2-(1-benzylpiperidin-4-yl)ethyl)-5,6-dihydroiso...)
Affinity DataIC50:  0.570nMAssay Description:In vitro inhibition of Acetylcholinesterase from human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50452874(CHEMBL4217620)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM312938(N-{2-[(4aR,6S,8aR)-2-amino-6-methyl-4,4a,5,6-tetra...)
Affinity DataIC50:  0.640nMAssay Description:Inhibition of BACE1 in human H4 cells transfected with wild type APP assessed as reduction in soluble portion of APPbeta level in cells incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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