Found 116 with Last Name = 'villarreal' and Initial = 'f' TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Agonist activity at FPR2 in human HL-60 cells assessed as reduction in chemoattractant induced chemotaxis by luminescence cell viability assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 0.00600nMAssay Description:Activation of eNOS in BCAEC assessed as increase in nitric oxide level after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Activation of eNOS in BCAEC assessed as increase in nitric oxide level after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Activation of eNOS in BCAEC assessed as increase in nitric oxide level after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A1/A2a/A2b/A3(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 6.17E+4nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A1/A2a/A2b/A3(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 5.13E+3nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A1/A2a/A2b/A3(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 6.76E+4nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
TargetAdenosine receptor A1/A2a/A2b/A3(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 8.71E+3nMAssay Description:Antagonist activity at Adenosine receptor in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional gentle stirri...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataEC50: 47nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at human FPR2 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human FPR1 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Agonist activity at mouse FPR2 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at mouse FPR1 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at human FPR2 expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: <1nMAssay Description:Agonist activity at FPR2 in mouse peritoneal macrophages assessed as inhibition of stimulated phagocytosis preincubated for 15 mins followed by FITC ...More data for this Ligand-Target Pair
Affinity DataEC50: 990nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 6.80nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.910nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.180nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 4.60nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 4.60nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.180nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0850nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.450nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
Affinity DataEC50: 3.10nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
