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Found 26 with Last Name = 'visy' and Initial = 'j'
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170230(CHEMBL445990)
Affinity DataIC50:  27nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460191(CHEMBL4225929)
Affinity DataIC50:  120nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460192(CHEMBL4224785)
Affinity DataIC50:  150nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246038((R)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-6(...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]SUC from succinic acid binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232880(Benzo[D]Isoxazol-3-Ol | CHEMBL444173)
Affinity DataIC50:  418nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246040((E,RS)-(6,7,8,9-tetrahydro-5-hydroxy-5H-benzocyclo...)
Affinity DataIC50:  500nMAssay Description:Displacement of [3H]SUC from succinic acid binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246038((R)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-6(...)
Affinity DataIC50:  800nMAssay Description:Displacement of [3H]GHB from gamma-hydroxybutyrate binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246040((E,RS)-(6,7,8,9-tetrahydro-5-hydroxy-5H-benzocyclo...)
Affinity DataIC50:  900nMAssay Description:Displacement of [3H]GHB from gamma-hydroxybutyrate binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460188(CHEMBL1886565)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22823(7-chloro-2,3-dihydro-1H-indole-2,3-dione | Isatin-...)
Affinity DataIC50:  7.87E+3nMAssay Description:Inhibition of DAAO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460189(CHEMBL4225931)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22821(7-methyl-2,3-dihydro-1H-indole-2,3-dione | Isatin-...)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of human DAAO using D-KYN as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by FP-6300-based flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246039((S,E)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-...)
Affinity DataIC50:  7.40E+4nMAssay Description:Displacement of [3H]SUC from succinic acid binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50246039((S,E)-2-(5-hydroxy-8,9-dihydro-5H-benzo[7]annulen-...)
Affinity DataIC50:  9.30E+4nMAssay Description:Displacement of [3H]GHB from gamma-hydroxybutyrate binding site of gamma-hydroxybutyrate receptor in rat forebrain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460194(CHEMBL2001613)
Affinity DataKd:  3.29E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460193(CHEMBL4227374)
Affinity DataKd:  780nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460192(CHEMBL4224785)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50232880(Benzo[D]Isoxazol-3-Ol | CHEMBL444173)
Affinity DataKd:  440nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50170230(CHEMBL445990)
Affinity DataKd:  870nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460189(CHEMBL4225931)
Affinity DataKd:  3.31E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460191(CHEMBL4225929)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460190(CHEMBL4225412)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM31148(3-hydroxyquinolin-2(1H)-one, 2 | US9701638, 1)
Affinity DataKd:  150nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM22821(7-methyl-2,3-dihydro-1H-indole-2,3-dione | Isatin-...)
Affinity DataKd:  8.23E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50460188(CHEMBL1886565)
Affinity DataKd:  4.59E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Sus scrofa (pig))
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50008990(1,2-Dihydro-indazol-3-one | 1H-indazol-3-ol | CHEM...)
Affinity DataKd:  4.43E+3nMAssay Description:Binding affinity to pig kidney DAAO by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed