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Found 30 with Last Name = 'wang' and Initial = 'ky'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50044625(CHEMBL3360190)
Affinity DataKi:  780nMAssay Description:Inhibition of CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Gilead Sciences

LigandPNGBDBM5244((5S,6S)-5-carbamimidamido-6-acetamido-1-(2-ethylbu...)
Affinity DataIC50:  140nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50144206((1S,2R,5S)-5-(6-Amino-purin-9-yl)-4-fluoro-3-hydro...)
Affinity DataIC50:  480nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50006222((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-hydroxymethyl-...)
Affinity DataIC50:  870nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50006215((1'R,2'S,3'R)-9-(2',3'-dihydroxycyclopent-4'-enyl)...)
Affinity DataIC50:  5.83E+3nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Gilead Sciences

LigandPNGBDBM5243((5S,6S)-5-amino-6-acetamido-1-(2-ethylbutanoyl)-1,...)
Affinity DataIC50:  6.00E+3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50144205((1S,2R,5S)-5-(6-Amino-purin-9-yl)-4-fluoro-cyclope...)
Affinity DataIC50:  7.67E+3nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50240464((S)-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)pe...)
Affinity DataIC50:  8.67E+3nMAssay Description:Antagonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus (B/Lee/40))
Gilead Sciences

LigandPNGBDBM5244((5S,6S)-5-carbamimidamido-6-acetamido-1-(2-ethylbu...)
Affinity DataIC50:  2.20E+4nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336547(5-(6-Aminopurin-9-yl)-4-chloro-3-hydroxymethylcycl...)
Affinity DataIC50:  3.65E+4nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336548(5-(6-Aminopurin-9-yl)-4-bromo-3-hydroxymethyl-cycl...)
Affinity DataIC50:  6.02E+4nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus (B/Lee/40))
Gilead Sciences

LigandPNGBDBM5243((5S,6S)-5-amino-6-acetamido-1-(2-ethylbutanoyl)-1,...)
Affinity DataIC50:  6.20E+4nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Gilead Sciences

LigandPNGBDBM5245((5R,6S)-5-amino-6-acetamido-1-(2-ethylbutanoyl)-1,...)
Affinity DataIC50:  1.60E+5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336551(5-(6-Aminopurin-9-yl)-4-bromocyclopent-3-ene-1,2-d...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336550(5-(6-Aminopurin-9-yl)-4-chlorocyclopent-3-ene-1,2-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus (B/Lee/40))
Gilead Sciences

LigandPNGBDBM5245((5R,6S)-5-amino-6-acetamido-1-(2-ethylbutanoyl)-1,...)
Affinity DataIC50: >1.00E+6nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336552(5-(6-Aminopurin-9-yl)-4-iodocyclopent-3-ene-1,2-di...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50336549(5-(6-Aminopurin-9-yl)-4-iodo-3-hydroxymethylcyclop...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human placental AdoHcy hydrolase expressed in Escherichia coli JM109More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataEC50:  4.13E+4nMAssay Description:Agonist activity at human recombinant PPARalpha expressed in HepG2 cells cotransfected with pGL3-PPRE3-TK-luc reporter assessed as beta-galactosidase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataKd:  32nMAssay Description:Binding affinity to human PPAR-alpha LBD assessed as recruitment of fluorescein-labeled coactivator peptide by surface plasmon resonance methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50044625(CHEMBL3360190)
Affinity DataKd:  1.93E+3nMAssay Description:Binding affinity to human PPAR-alpha LBD assessed as recruitment of fluorescein-labeled coactivator peptide by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50:  4.50E+3nMAssay Description:Binding affinity to histidine-tagged human PPARalpha-LBD assessed as recruitment of co-activator peptide fluorescein-labeled PGC1alpha after 2 hrs by...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50044625(CHEMBL3360190)
Affinity DataEC50:  9.58E+3nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataKd:  9.64E+4nMAssay Description:Binding affinity to PPARalpha LBD (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50240464((S)-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)pe...)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to PPARalpha LBD (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  1.86E+4nMAssay Description:Agonist activity at PPARalpha LBD (unknown origin) assessed as induction of PGC1alpha co-activator activity by TR-FRET analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50240464((S)-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)pe...)
Affinity DataEC50:  8.34E+4nMAssay Description:Agonist activity at PPARalpha LBD (unknown origin) assessed as induction of PGC1alpha co-activator activity by TR-FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50044625(CHEMBL3360190)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at PPAR-alpha (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed