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Found 199 with Last Name = 'watt' and Initial = 'k'
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM185171(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataKi:  150nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM61867(2-(4-hydroxyphenyl)-5,6,7,8-tetrakis(oxidanyl)chro...)
Affinity DataKi:  1.29E+3nMAssay Description:Competitive inhibition of PFKFB3 (unknown origin) using fructose 6-phosphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataKi:  1.49E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608169(CHEMBL5290129)
Affinity DataKi:  1.95E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608171(CHEMBL5268027)
Affinity DataKi:  2.32E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataKi:  3.98E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589238(CHEMBL5185481)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589244(CHEMBL5176597)
Affinity DataKi:  6.51E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608174(CHEMBL5291124)
Affinity DataKi:  8.83E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589233(CHEMBL5199766)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608175(CHEMBL5269953)
Affinity DataKi:  2.63E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589243(CHEMBL5174050)
Affinity DataKi:  2.74E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608170(CHEMBL5278364)
Affinity DataKi:  3.06E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589239(CHEMBL5183970)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608167(CHEMBL5276215)
Affinity DataKi:  3.84E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589242(CHEMBL5180097)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589234(CHEMBL5203769)
Affinity DataKi:  5.16E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608168(CHEMBL5266611)
Affinity DataKi:  6.18E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589240(CHEMBL5169952)
Affinity DataKi:  6.45E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608172(CHEMBL5269861)
Affinity DataKi:  7.01E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589241(CHEMBL5171356)
Affinity DataKi:  7.42E+4nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608173(CHEMBL5282572)
Affinity DataKi:  8.85E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589237(CHEMBL5196710)
Affinity DataKi:  1.09E+5nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589235(CHEMBL5177045)
Affinity DataKi:  1.34E+5nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50589236(CHEMBL5188696)
Affinity DataKi:  1.42E+5nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608176(CHEMBL5270888)
Affinity DataKi:  1.54E+5nMAssay Description:Reversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50073654(4-(Methylsulfinyl)Butyl Isothiocyanate | CHEBI:478...)
Affinity DataKi:  3.66E+5nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567964(CHEMBL4858336 | US11903936, Compound 29)
Affinity DataIC50:  12nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567964(CHEMBL4858336 | US11903936, Compound 29)
Affinity DataIC50:  25nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50365230(CHEMBL1956285 | US11903936, Compound DSM265 | US92...)
Affinity DataIC50:  30nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567990(CHEMBL4846297 | US11903936, Compound 8)
Affinity DataIC50:  32nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567990(CHEMBL4846297 | US11903936, Compound 8)
Affinity DataIC50:  34nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567995(CHEMBL4851471 | US11903936, Compound 20)
Affinity DataIC50:  41nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567967(CHEMBL4850393 | US11903936, Compound 35)
Affinity DataIC50:  41nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567992(CHEMBL4846204 | US11903936, Compound 11)
Affinity DataIC50:  41nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567994(CHEMBL4864218 | US11903936, Compound 17)
Affinity DataIC50:  43nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM651975(3-methyl-N-(1-(1H-pyrazol-4-yl)ethyl)-4-(((trifluo...)
Affinity DataIC50:  43nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM651975(3-methyl-N-(1-(1H-pyrazol-4-yl)ethyl)-4-(((trifluo...)
Affinity DataIC50:  47nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567967(CHEMBL4850393 | US11903936, Compound 35)
Affinity DataIC50:  50nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567991(CHEMBL4848632 | US11903936, Compound 2)
Affinity DataIC50:  52nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567992(CHEMBL4846204 | US11903936, Compound 11)
Affinity DataIC50:  57nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM651960(N-(1-(1H-1,2,4-triazol-3-yl) ethyl)-4-(3-fluoro-4-...)
Affinity DataIC50:  61nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50365230(CHEMBL1956285 | US11903936, Compound DSM265 | US92...)
Affinity DataIC50:  72nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(malaria parasite P. vivax)
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567998(CHEMBL4876457 | US11903936, Compound 26)
Affinity DataIC50:  74nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567995(CHEMBL4851471 | US11903936, Compound 20)
Affinity DataIC50:  76nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567994(CHEMBL4864218 | US11903936, Compound 17)
Affinity DataIC50:  85nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Mahidol University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human VEGFR2 kinase domain expressed in SF9 cells by TR-FRET assayMore data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567998(CHEMBL4876457 | US11903936, Compound 26)
Affinity DataIC50:  96nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Plasmodium falciparum (isolate 3D7))
The Board of Regents of The University of Texas System

US Patent
LigandPNGBDBM50567991(CHEMBL4848632 | US11903936, Compound 2)
Affinity DataIC50:  98nMAssay Description:The 50% inhibitory concentration (IC50) for the described compounds was determined using the 2,6-dichloroindophenol (DCIP) assay to monitor the DHODH...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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