Found 3 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM185173' TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Inhibition of recombinant human TG2 expressed in Escherichia coli assessed as inhibition constant using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) a...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University Of Ottawa
Curated by ChEMBL
University Of Ottawa
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
