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Found 436 with Last Name = 'watts' and Initial = 'vj'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094670(1-(4-Dipropylamino-1,3,4,5-tetrahydro-benzo[cd]ind...)
Affinity DataKi:  0.0880nMAssay Description:Inhibition constant of 50 microM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50004822((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity towards dopamine receptor D1 using [3H]-SCH-23,390 was determined in rat striatal membranesChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  0.920nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.940nMAssay Description:Displacement of [3H]-SCH-23390 from human dopamine D1 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50394089(CHEMBL2158640)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D2long receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD1 dopamine receptor(Monkey)
University of North Carolina

Curated by PDSP Ki Database
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(CHEMBL342986 | Diethyl-[2-(5-methoxy-1H-indol-3-yl...)
Affinity DataKi:  1.70nMAssay Description:Evaluated for the binding constant at [3H]-8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200351((+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chrom...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human cloned adrenergic alpha 2C receptor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  5.40nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50117181((S)-2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinol...)
Affinity DataKi:  5.93nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50038349((S)-6-Chloro-2-methyl-1-phenyl-1,2,3,4-tetrahydro-...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity towards dopamine receptor D1 using [3H]-SCH-23,390 was determined in rat striatal membranesChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50038349((S)-6-Chloro-2-methyl-1-phenyl-1,2,3,4-tetrahydro-...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity towards dopamine receptor D1 using [3H]-SCH-23,390 was determined in rat striatal membranesChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50020222((+/-)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200351((+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chrom...)
Affinity DataKi:  7nMAssay Description:Binding affinity to human cloned dopamine D5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094671(3-(2-Dimethylamino-ethyl)-6-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  7.40nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200353((6aR,12bS)-(+)-2,3-dihydroxy-6a,7,8,12b-tetrahydro...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]spiperone from dopamine D2-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50038345((S)-6-Bromo-2-methyl-1-phenyl-1,2,3,4-tetrahydro-i...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity towards dopamine receptor D1 using [3H]-SCH-23,390 was determined in rat striatal membranesChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50032522((6aR,12bS)-2-Methyl-5,6,6a,7,8,12b-hexahydro-benzo...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  10nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200351((+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chrom...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human cloned adrenergic alpha 2B receptor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  13nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(CHEMBL342986 | Diethyl-[2-(5-methoxy-1H-indol-3-yl...)
Affinity DataKi:  16nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  16.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669(CHEMBL337590 | [2-(6-Fluoro-5-methoxy-1H-indol-3-y...)
Affinity DataKi:  19nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD1 dopamine receptor(Monkey)
University of North Carolina

Curated by PDSP Ki Database
LigandPNGBDBM50010685((+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahyd...)
Affinity DataKi:  20.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50200351((+/-)-2,3-dihydroxy-6a,7,8,12b-tetrahydro-6H-chrom...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1-like receptor in porcine striata homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  25nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50032517((6aR,12bS)-2-Ethyl-5,6,6a,7,8,12b-hexahydro-benzo[...)
Affinity DataKi:  29nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50117181((S)-2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinol...)
Affinity DataKi:  31.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669(CHEMBL337590 | [2-(6-Fluoro-5-methoxy-1H-indol-3-y...)
Affinity DataKi:  33nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50004822((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)
Affinity DataKi:  41.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(CHEMBL342986 | Diethyl-[2-(5-methoxy-1H-indol-3-yl...)
Affinity DataKi:  42nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50010685((+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahyd...)
Affinity DataKi:  43.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-SCH-23390 from human dopamine D1 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(CHEMBL142936 | Diethyl-[2-(1H-indol-3-yl)-ethyl]-a...)
Affinity DataKi:  47nMAssay Description:Evaluated for the binding constant at [3H]-8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  49nMAssay Description:Evaluated for the binding constant at [3H]-8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50394091(CHEMBL2158636)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Purdue University

Curated by PDSP Ki Database
LigandPNGBDBM50022052(1-Benzyl-6-chloro-2-methyl-1,2,3,4-tetrahydro-isoq...)
Affinity DataKi:  53nMAssay Description:Binding affinity of compound towards dopamine (D1) receptor using [3H]-SCH-23,390 was determined in rat striatal membranesChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094674(CHEMBL142862 | [2-(4-Fluoro-5-methoxy-1H-indol-3-y...)
Affinity DataKi:  55nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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