Affinity DataKi: 230nMAssay Description:Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human HEK293T cells after 45 mins by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in HEK293T cells after 1 hr by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKd: 76nMAssay Description:Binding affinity to NF-kappaB p50 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+4nMAssay Description:Binding affinity to NF-kappaB RelA (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.34E+3nMAssay Description:Binding affinity to NF-kappaB RelA (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKd: 216nMAssay Description:Binding affinity to NF-kappaB p50 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair