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Found 21 with Last Name = 'weerapana' and Initial = 'e'
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Pfizer

LigandPNGBDBM81356(PF-3845, 10)
Affinity DataKi:  230nMAssay Description:Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Pfizer

LigandPNGBDBM26739(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Affinity DataKi:  2.00E+3nMAssay Description:Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM75707((3R)-3-cyclopentyl-4-keto-3-phenyl-diazetidine-1,2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human HEK293T cells after 45 mins by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400987(CHEMBL1316687)
Affinity DataIC50:  640nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400996(CHEMBL1699083)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400995(CHEMBL1706554)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400994(CHEMBL1719837)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400988(CHEMBL1701914)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in HEK293T cells after 1 hr by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400993(CHEMBL1729870)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400989(CHEMBL1718102)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400991(CHEMBL1711185)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400997(CHEMBL1521288)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400990(CHEMBL1723004)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400992(CHEMBL1701983)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50561593(CHEBI:2598 | CHEMBL2359602)
Affinity DataKd:  76nMAssay Description:Binding affinity to NF-kappaB p50 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50561592((+)-Gibberellic Acid | CHEBI:28833 | GIBBERELLIN A...)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to NF-kappaB RelA (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50561593(CHEBI:2598 | CHEMBL2359602)
Affinity DataKd:  6.34E+3nMAssay Description:Binding affinity to NF-kappaB RelA (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50561592((+)-Gibberellic Acid | CHEBI:28833 | GIBBERELLIN A...)
Affinity DataKd:  216nMAssay Description:Binding affinity to NF-kappaB p50 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed