Affinity DataIC50: 120nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.12E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.12E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.86E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.86E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.26E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.26E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 9.26E+3nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.86E+3nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of electric eel AChE by modified Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of human acetyl cholinesterase by Ellmann's methodMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.51E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.59E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 4.91E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.28E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.29E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.61E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.81E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 5.84E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged SIRT1 (193 to 741 amino acid) after 45 mins by spectrophotometry relative to controlMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human recombinant C-terminal His-tagged SIRT2 (13 to 319) after 45 mins by fluorescence assayMore data for this Ligand-Target Pair