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Found 177 with Last Name = 'weigelt' and Initial = 't'
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136352(US8859534, 38)
Affinity DataKi:  0.0640nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136326(US8859534, 12)
Affinity DataKi:  0.110nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136317(US8859534, 3)
Affinity DataKi:  0.140nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136354(US8859534, 40)
Affinity DataKi:  0.140nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136363(US8859534, 49)
Affinity DataKi:  0.160nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136362(US8859534, 48)
Affinity DataKi:  0.160nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136325(US8859534, 11)
Affinity DataKi:  0.160nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136318(US8859534, 4)
Affinity DataKi:  0.200nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397757(CHEMBL2177173)
Affinity DataKi:  0.220nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136361(US8859534, 47)
Affinity DataKi:  0.220nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136351(US8859534, 37)
Affinity DataKi:  0.230nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136365(US8859534, 51)
Affinity DataKi:  0.230nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136322(US8859534, 8)
Affinity DataKi:  0.280nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136322(US8859534, 8)
Affinity DataKi:  0.290nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136353(US8859534, 39)
Affinity DataKi:  0.320nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136357(US8859534, 43)
Affinity DataKi:  0.330nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136359(US8859534, 45)
Affinity DataKi:  0.340nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136367(US8859534, 53)
Affinity DataKi:  0.350nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136324(US8859534, 10)
Affinity DataKi:  0.380nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397744(CHEMBL2177163)
Affinity DataKi:  0.400nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136338(US8859534, 24)
Affinity DataKi:  0.420nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136364(US8859534, 50)
Affinity DataKi:  0.430nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136323(US8859534, 9)
Affinity DataKi:  0.440nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136350(US8859534, 36)
Affinity DataKi:  0.460nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397749(CHEMBL2182002)
Affinity DataKi:  0.460nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397756(CHEMBL2177174)
Affinity DataKi:  0.480nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136317(US8859534, 3)
Affinity DataKi:  0.520nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136327(US8859534, 13)
Affinity DataKi:  0.550nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136338(US8859534, 24)
Affinity DataKi:  0.560nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136321(US8859534, 7)
Affinity DataKi:  0.590nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136356(US8859534, 42)
Affinity DataKi:  0.640nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397743(CHEMBL2177165)
Affinity DataKi:  0.670nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136332(US8859534, 18)
Affinity DataKi:  0.700nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136330(US8859534, 16)
Affinity DataKi:  0.780nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136342(US8859534, 28)
Affinity DataKi:  0.850nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136326(US8859534, 12)
Affinity DataKi:  0.880nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136324(US8859534, 10)
Affinity DataKi:  0.890nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136340(US8859534, 26)
Affinity DataKi:  0.910nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136336(US8859534, 22)
Affinity DataKi:  0.910nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136333(US8859534, 19)
Affinity DataKi:  0.990nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397753(CHEMBL2177177)
Affinity DataKi:  0.990nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136342(US8859534, 28)
Affinity DataKi:  1nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50397748(CHEMBL2177155)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human recombinant GSK3beta using biotin- AAEELDSRAGS(PO3H2)PQL as substrate and [gamma32P]ATP after 20 mins by scintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136344(US8859534, 30)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136334(US8859534, 20)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136316(US8859534, 2)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1B(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136354(US8859534, 40)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136355(US8859534, 41)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136315(US8859534, 1)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Cricetulus griseus (Chinese hamster) (Cricetulus b...)
Acturum Life Science

US Patent
LigandPNGBDBM136360(US8859534, 46)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:Assays that were used to measure affinity of the compounds of the present invention for 5-HT1A and 5-HT1B receptors are described in J. Recept Signal...More data for this Ligand-Target Pair
In DepthDetails US Patent
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