Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Wyeth Research
Curated by ChEMBL
Wyeth Research
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human Tpl2 by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Wyeth Research
Curated by ChEMBL
Wyeth Research
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human Tpl2 by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAlpha-mannosidase 2C1(Rattus norvegicus)
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Csiro Division Of Chemicals And Polymers
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibitory activity against Mannosidase in jack bean (Canavalia ensiformis)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of IL-1-beta-stimulated MMP3 in human RA-FLS cells by immunoblot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonist activity at alpha4beta1 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at N-cadherinMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.25E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.75E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Binding affinity to N-terminal thioredoxin-His6 tag with N-terminal thrombin-cleavage site containing recombinant BCL6 BTB domain C8Q/C67R/C84N/E99V ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Wyeth Research
Curated by ChEMBL
Wyeth Research
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human Tpl2 by ELISAMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Oryctolagus cuniculus (rabbit))
Wyeth Research
Curated by ChEMBL
Wyeth Research
Curated by ChEMBL
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of rabbit MEK1 by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of human EGFR by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+4nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair