Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: >9.30E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >9.30E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
Affinity DataEC50: 770nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0630nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.05E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.75E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair