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Found 81 with Last Name = 'winssinger' and Initial = 'n'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557999(CHEMBL4786214)
Affinity DataKi:  250nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557998(CHEMBL4796866)
Affinity DataKi:  250nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557984(CHEMBL4744734)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557985(CHEMBL4759705)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557997(CHEMBL4786563)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557996(CHEMBL4778692)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557995(CHEMBL4800222)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557994(CHEMBL4793855)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557988(CHEMBL4786891)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557989(CHEMBL4779255)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557987(CHEMBL4777832)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557986(CHEMBL4746426)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557981(CHEMBL4796812)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557980(CHEMBL4741877)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557983(CHEMBL4793211)
Affinity DataKi:  3.01E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557982(CHEMBL4762824)
Affinity DataKi:  3.01E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557990(CHEMBL4752726)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557991(CHEMBL4754600)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557985(CHEMBL4759705)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557984(CHEMBL4744734)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557992(CHEMBL4762078)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557993(CHEMBL4740579)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557992(CHEMBL4762078)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557993(CHEMBL4740579)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557983(CHEMBL4793211)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557982(CHEMBL4762824)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557980(CHEMBL4741877)
Affinity DataKi:  7.01E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557981(CHEMBL4796812)
Affinity DataKi:  7.01E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557988(CHEMBL4786891)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557989(CHEMBL4779255)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557990(CHEMBL4752726)
Affinity DataKi:  1.22E+4nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557991(CHEMBL4754600)
Affinity DataKi:  1.22E+4nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557987(CHEMBL4777832)
Affinity DataKi:  1.68E+4nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557986(CHEMBL4746426)
Affinity DataKi:  1.68E+4nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human PTP1B (1 to 321 residues) expressed in Escherichia coli using DifMup as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557998(CHEMBL4796866)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557999(CHEMBL4786214)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557997(CHEMBL4786563)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557996(CHEMBL4778692)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557995(CHEMBL4800222)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50557994(CHEMBL4793855)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of recombinant human TCPTP (1 to 317 residues) expressed in Escherichia coli using DifMup as substrate preincubated for 30 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341234(4-(chloromethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)py...)
Affinity DataIC50:  139nMAssay Description:Inhibition of human wild type PDGFRalpha assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human wild type PDGFRalpha assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341234(4-(chloromethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)py...)
Affinity DataIC50:  245nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341235(4-(aminomethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyr...)
Affinity DataIC50:  788nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341236(4-((2-chloroacetamido)methyl)-N-(4-methyl-3-(4-(py...)
Affinity DataIC50:  788nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341236(4-((2-chloroacetamido)methyl)-N-(4-methyl-3-(4-(py...)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of human wild type PDGFRalpha assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341235(4-(aminomethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyr...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human wild type PDGFRalpha assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human wild type ABL1 assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341238(4-(methacrylamidomethyl)-N-(4-methyl-3-(4-(pyridin...)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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