TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibition of recombinant N-terminal FLAG-tagged FAP (unknown origin) (38 to 760 residues) expressed in HEK293 cells using AMCC as substrate by fluor...More data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate measured upto 60 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 663nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 7.98E+4nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 8.53E+4nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 1.47E+6nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 1(Rattus norvegicus)
Peking University First Hospital
Curated by ChEMBL
Peking University First Hospital
Curated by ChEMBL
Affinity DataIC50: 1.72E+6nMAssay Description:Inhibition of FAP in human U87MG cells using Suc-Gly-Pro-AMC as substrate by fluorescence based assayMore data for this Ligand-Target Pair