TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Competitive inhibition of human full-length recombinant HDAC6 expressed in baculovirus infected Sf9 insect cells using Boc-Lys (Ac)-AMC as substrate ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of Escherichia coli DHFRMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory activity against beta-1 adrenergic receptor determined as pA2 in guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of human full-length recombinant HDAC6 expressed in baculovirus infected Sf9 insect cells using Boc-Lys (Ac)-AMC as substrate preincubated...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 2.60nMAssay Description:Inhibition of human HDAC6 CD2 expressed in Escherichia coli BL21 (RIL) using Boc-Lys (Ac)-AMC as substrate preincubated for 10 mins followed by subst...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of human full-length recombinant HDAC6 expressed in baculovirus infected Sf9 insect cells using Boc-Lys (Ac)-AMC as substrate preincubated...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Competitive inhibition of human HDAC6 CD2 expressed in Escherichia coli BL21 (RIL) using Boc-Lys (Ac)-AMC as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of human full-length recombinant HDAC6 expressed in baculovirus infected Sf9 insect cells using Boc-Lys (Ac)-AMC as substrate preincubated...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of wild type Staphylococcus aureus DHFRMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.5nMAssay Description:Inhibition of human HDAC6 CD2 expressed in Escherichia coli BL21 (RIL) using Boc-Lys (Ac)-AMC as substrate preincubated for 10 mins followed by subst...More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Inhibition of Escherichia coli DHFR assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 9.40nMAssay Description:In vitro inhibitory activity against beta-1 adrenergic receptor determined as pA2 in guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro inhibitory activity against beta-1 adrenergic receptor determined as pA2 in guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of 25-[26,27-3H]hydroxycholesterol from RORgammat receptor ligand binding domain (unknown origin) after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 32nMAssay Description:Displacement of 25-[26,27-3H]hydroxycholesterol from RORgammat receptor ligand binding domain (unknown origin) after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of 25-[26,27-3H]hydroxycholesterol from RORgammat receptor ligand binding domain (unknown origin) after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 191nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 120 nMMore data for this Ligand-Target Pair
Affinity DataKi: 203nMAssay Description:Compound was tested for the inhibition of chymotrypsin at 69 nMMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database