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Found 652 with Last Name = 'van den berg' and Initial = 'rj'
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376888(CHEMBL415279)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376892(CHEMBL406958)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376889(CHEMBL260647)
Affinity DataKi:  260nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376893(CHEMBL262334)
Affinity DataKi:  380nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376878(CHEMBL436906)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376877(CHEMBL259878)
Affinity DataKi:  480nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376883(CHEMBL404611)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376873(CHEMBL438168)
Affinity DataKi:  510nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376896(CHEMBL262599)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376890(CHEMBL261649)
Affinity DataKi:  580nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376895(CHEMBL406960)
Affinity DataKi:  600nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376875(CHEMBL260812)
Affinity DataKi:  620nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376899(CHEMBL260318)
Affinity DataKi:  700nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376876(CHEMBL408760)
Affinity DataKi:  720nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376874(CHEMBL260750)
Affinity DataKi:  740nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376891(CHEMBL439076)
Affinity DataKi:  770nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376880(CHEMBL436862)
Affinity DataKi:  820nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376885(CHEMBL262335)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376884(CHEMBL429690)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376897(CHEMBL406084)
Affinity DataKi:  930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376879(CHEMBL266172)
Affinity DataKi:  930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376900(CHEMBL258970)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376898(CHEMBL408759)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376894(CHEMBL259220)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376881(CHEMBL406713)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376887(CHEMBL436878)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376886(CHEMBL436697)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376882(CHEMBL437260)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028180(CHEMBL3354625)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028244(CHEMBL3354627)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028179(CHEMBL3354624)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028255(CHEMBL3354635)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028254(CHEMBL3354634)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028181(CHEMBL3354626)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028256(CHEMBL3354636)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028221(CHEMBL3354041)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028257(CHEMBL3354637)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Mus musculus)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211257(CHEMBL3895863 | US10583137, Compound 14)
Affinity DataIC50:  0.631nMAssay Description:Inhibition of MB064 probe binding to DAGLalpha in mouse brain membrane proteome preincubated for 30 mins followed by MB064 probe addition measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211240(CHEMBL3897587)
Affinity DataIC50:  0.631nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in HEK293T cell membranes overexpressing MAGL using natural substrate 1-stearoyl-2-arachidonoly-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211265(CHEMBL3954476)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in HEK293T cell membranes overexpressing MAGL using natural substrate 1-stearoyl-2-arachidonoly-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211266(CHEMBL3906477)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of full length recombinant human DAGLalpha expressed in HEK293T cell membranes using PNP butyrate as substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211271(CHEMBL3913807)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in HEK293T cell membranes overexpressing MAGL using natural substrate 1-stearoyl-2-arachidonoly-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028203(CHEMBL3354021)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028204(CHEMBL3354022)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028229(CHEMBL3354048)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50312527(CHEMBL1086996 | N-[5-(Adamantan-1-yl-methoxy)-pent...)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028230(CHEMBL3354049)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50312529(CHEMBL1088158 | N-[5-(Adamantan-1-yl-methoxy)-pent...)
Affinity DataIC50: <1nMAssay Description:Inhibition of GBA2 by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50028215(CHEMBL3354035)
Affinity DataIC50:  1nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50312527(CHEMBL1086996 | N-[5-(Adamantan-1-yl-methoxy)-pent...)
Affinity DataIC50: <1nMAssay Description:Inhibition of GBA2 by HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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