TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 794nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 6.31E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 7.94E+5nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
Affinity DataIC50: 274nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair