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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
467
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
Ki: 26nM
Assay Description:
Inhibitory activity against VEGFR2
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 26nM
Assay Description:
Inhibitory activity against VEGFR2
More data for this Ligand-Target Pair
Target Info
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MMDB
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Target
Vascular endothelial growth factor receptor 2
(Mus musculus)
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 28nM
Assay Description:
Inhibitory activity against Flk1
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 60nM
Assay Description:
Inhibitory activity against VEGFR1
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 25nM
Assay Description:
Inhibition of human VEGFR2
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 26nM
Assay Description:
Inhibition of human recombinant VEGFR-2
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 26nM
Assay Description:
Inhibition of recombinant VEGFR-2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: 28nM
Assay Description:
Inhibition of recombinant FGFR-1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: 28nM
Assay Description:
Inhibition of human recombinant FGFR-1
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 2
(Mus musculus)
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: 89nM
Assay Description:
Inhibitory activity against Flk1
More data for this Ligand-Target Pair
Target Info
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: 148nM
Assay Description:
Inhibitory activity against FGFR1
More data for this Ligand-Target Pair
Target Info
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 380nM
Assay Description:
Inhibitory activity against VEGFR1
More data for this Ligand-Target Pair
Target Info
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >1.90E+3nM
Assay Description:
Inhibitory activity against EGFR
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: >2.50E+3nM
Assay Description:
Inhibitory activity against LCK
More data for this Ligand-Target Pair
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Target
Platelet-derived growth factor receptor beta
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >6.00E+3nM
Assay Description:
Inhibitory activity against PDGFRbeta
More data for this Ligand-Target Pair
Target Info
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: 1.80E+4nM
Assay Description:
Inhibitory activity against hERG by patch-clamp assay
More data for this Ligand-Target Pair
Target Info
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Target
Cytochrome P450 3A4
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: 1.80E+4nM
Assay Description:
Inhibition of human CYP3A4 using 7-benzyl-trifluoromethyl coumarin
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Cytochrome P450 3A4
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.80E+4nM
Assay Description:
Inhibitory activity against CYP3A4
More data for this Ligand-Target Pair
Target Info
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Target
Protein kinase C alpha type
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibitory activity against PKC alpha
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Cytochrome P450 2D6
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: >4.00E+4nM
Assay Description:
Inhibition of human CYP2D6
More data for this Ligand-Target Pair
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Target
Cytochrome P450 2C9
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >4.00E+4nM
Assay Description:
Inhibition of human CYP2C9
More data for this Ligand-Target Pair
Target Info
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Target
Cytochrome P450 1A2
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >4.00E+4nM
Assay Description:
Inhibition of human CYP1A2
More data for this Ligand-Target Pair
Target Info
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Target
Cytochrome P450 3A4
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: 4.00E+4nM
Assay Description:
Inhibition of human CYP3A4 using 7-benzyloxyresorufin
More data for this Ligand-Target Pair
Target Info
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Target
Cytochrome P450 2C19
(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
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Affinity Data
IC50: >4.00E+4nM
Assay Description:
Inhibition of human CYP2C19
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase JAK3
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibitory activity against JAK3
More data for this Ligand-Target Pair
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 640nM
Assay Description:
Binding constant for ABL1(H396P)-phosphorylated kinase domain
More data for this Ligand-Target Pair
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Target
Ephrin type-A receptor 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA1 kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(S752-I759del) kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 450nM
Assay Description:
Binding constant for ABL1(M351T)-phosphorylated kinase domain
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Target
Insulin receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for INSR kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.10E+3nM
Assay Description:
Binding constant for ABL1(Y253F)-phosphorylated kinase domain
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(D835Y) kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 580nM
Assay Description:
Binding constant for ABL1(E255K)-phosphorylated kinase domain
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 390nM
Assay Description:
Binding constant for ABL1(H396P)-nonphosphorylated kinase domain
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Copy BDB DOI
Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(ITD) kinase domain
More data for this Ligand-Target Pair
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Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 150nM
Assay Description:
Binding constant for FGFR3(G697C) kinase domain
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Target
eIF-2-alpha kinase GCN2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for GCN2(Kin.Dom.2,S808G) kinase domain
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Target
Serine/threonine-protein kinase MRCK gamma
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DMPK2 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(H1047L) kinase domain
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Target
Ribosomal protein S6 kinase alpha-5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RPS6KA5(Kin.Dom.1-N-terminal) kinase domain
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Target Info
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Target
Myosin light chain kinase, smooth muscle
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MYLK kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 17nM
Assay Description:
Binding constant for KIT(V559D,T670I) kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.20E+3nM
Assay Description:
Binding constant for ABL1(Q252H)-phosphorylated kinase domain
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Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RET(V804M) kinase domain
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Target
Non-receptor tyrosine-protein kinase TYK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TYK2(JH2domain-pseudokinase) kinase domain
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Target
Protein kinase C eta type
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKCH kinase domain
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Target
Macrophage-stimulating protein receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MST1R kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 3.00E+3nM
Assay Description:
Binding constant for EGFR(G719C) kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Calcium/calmodulin-dependent protein kinase type II subunit alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK2A kinase domain
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Target
Serine/threonine-protein kinase Chk1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CHEK1 kinase domain
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Target
Death-associated protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DAPK1 kinase domain
More data for this Ligand-Target Pair
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Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 360nM
Assay Description:
Binding constant for RET(M918T) kinase domain
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Target
MAP/microtubule affinity-regulating kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MARK3 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(E545K) kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(K663Q) kinase domain
More data for this Ligand-Target Pair
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Target
Serine/threonine-protein kinase 17A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DRAK1 kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(L747-S752del, P753S) kinase domain
More data for this Ligand-Target Pair
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.70E+3nM
Assay Description:
Binding constant for ABL1(T315I)-nonphosphorylated kinase domain
More data for this Ligand-Target Pair
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(L858R,T790M) kinase domain
More data for this Ligand-Target Pair
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Target
SRSF protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SRPK2 kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(T790M) kinase domain
More data for this Ligand-Target Pair
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Target
Serine/threonine-protein kinase B-raf
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BRAF kinase domain
More data for this Ligand-Target Pair
Target Info
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NCI pathway
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 4.00E+3nM
Assay Description:
Binding constant for KIT(D816V) kinase domain
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Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AAK1 kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.10E+3nM
Assay Description:
Binding constant for ABL1-nonphosphorylated kinase domain
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Target
Myosin-IIIb
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MYO3B kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(L747-E749del, A750P) kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for KIT(A829P) kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(M1043I) kinase domain
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Target
Cyclin-dependent kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK4-cyclinD1 kinase domain
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Target Info
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(E545A) kinase domain
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(D835H) kinase domain
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Target
Serine/threonine-protein kinase D2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKD2 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(C420R) kinase domain
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Target
Calcium/calmodulin-dependent protein kinase kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMKK2 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(I800L) kinase domain
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Target
Ribosomal protein S6 kinase alpha-6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK4(Kin.Dom.2-C-terminal) kinase domain
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Target
Aurora kinase B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AURKB kinase domain
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Target
Interleukin-1 receptor-associated kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for IRAK3 kinase domain
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Target
cGMP-dependent protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKG1 kinase domain
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Target
Ribosomal protein S6 kinase alpha-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK3(Kin.Dom.1-N-terminal) kinase domain
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MET kinase domain
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Target
Rho-associated protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ROCK2 kinase domain
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Target
Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 56nM
Assay Description:
Binding constant for FLT4 kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 4.10E+3nM
Assay Description:
Binding constant for ABL1(F317L)-nonphosphorylated kinase domain
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Target
Ephrin type-A receptor 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 190nM
Assay Description:
Binding constant for EPHA6 kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(E746-A750del) kinase domain
More data for this Ligand-Target Pair
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Target
Mitogen-activated protein kinase kinase kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP3K4 kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for KIT(D816H) kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type II subunit beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK2B kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(Q546K) kinase domain
More data for this Ligand-Target Pair
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Target
Serine/threonine-protein kinase BRSK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BRSK1 kinase domain
More data for this Ligand-Target Pair
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ABL1(F317I)-nonphosphorylated kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 2.60E+3nM
Assay Description:
Binding constant for EGFR(G719S) kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ABL1(F317I)-phosphorylated kinase domain
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Target
Leucine-rich repeat serine/threonine-protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for LRRK2(G2019S) kinase domain
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Target
Cyclin-dependent kinase 11A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDC2L2 kinase domain
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Target
Ribosomal protein S6 kinase alpha-4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RPS6KA4(Kin.Dom.2-C-terminal) kinase domain
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Target Info
NCI pathway
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 54nM
Assay Description:
Binding constant for KIT(L576P) kinase domain
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Target
Myotonin-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DMPK kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.50E+3nM
Assay Description:
Binding constant for ABL1(Q252H)-nonphosphorylated kinase domain
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Target
Ribosomal protein S6 kinase alpha-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK1(Kin.Dom.2-C-terminal) kinase domain
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Target Info
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 12nM
Assay Description:
Binding constant for KIT(V559D,V654A) kinase domain
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Target
Misshapen-like kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 310nM
Assay Description:
Binding constant for MINK kinase domain
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Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for RET(V804L) kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 640nM
Assay Description:
Binding constant for ABL1-phosphorylated kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 5.10E+3nM
Assay Description:
Binding constant for EGFR(L858R) kinase domain
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Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JAK1(JH2domain-pseudokinase) kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 36nM
Assay Description:
Binding constant for KIT kinase domain
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Target
Inhibitor of nuclear factor kappa-B kinase subunit alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for IKK-alpha kinase domain
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MET(Y1235D) kinase domain
More data for this Ligand-Target Pair
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EGFR(L747-T751del,Sins) kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(N841I) kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(E542K) kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 450nM
Assay Description:
Binding constant for ABL1(T315I)-phosphorylated kinase domain
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Target
Serine/threonine-protein kinase TNNI3K
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TNNI3K kinase domain
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Target
Cyclin-dependent kinase 15
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PFTAIRE2 kinase domain
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Target
Rhodopsin kinase GRK7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for GRK7 kinase domain
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Target Info
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Target
Homeodomain-interacting protein kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for HIPK4 kinase domain
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Target
Dual specificity mitogen-activated protein kinase kinase 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 3.10E+3nM
Assay Description:
Binding constant for MEK5 kinase domain
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Target
Dual specificity mitogen-activated protein kinase kinase 7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MKK7 kinase domain
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Target
Casein kinase I isoform alpha-like
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1A1L kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TAK1 kinase domain
More data for this Ligand-Target Pair
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Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 590nM
Assay Description:
Binding constant for MAP4K4 kinase domain
More data for this Ligand-Target Pair
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Target
Serine/threonine-protein kinase Nek11
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK11 kinase domain
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Target
Homeodomain-interacting protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for HIPK1 kinase domain
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Target
Tyrosine-protein kinase Fyn
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FYN kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Serine/threonine-protein kinase NIM1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NIM1 kinase domain
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Target Info
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Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FAK kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type II subunit gamma
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK2G kinase domain
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Target
Protein-tyrosine kinase 2-beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PYK2 kinase domain
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Target
Serine/threonine-protein kinase SIK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SIK kinase domain
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Target Info
NCI pathway
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Target
Serine/threonine-protein kinase 32C
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for YANK3 kinase domain
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Target
Ankyrin repeat and protein kinase domain-containing protein 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ANKK1 kinase domain
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Target
Ephrin type-A receptor 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA5 kinase domain
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Target Info
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Target
Myosin light chain kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MLCK kinase domain
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Target
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKMYT1 kinase domain
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Target
G protein-coupled receptor kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for GRK4 kinase domain
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Target
Leucine-rich repeat serine/threonine-protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LRRK2 kinase domain
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Target
Serine/threonine-protein kinase Nek5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK5 kinase domain
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Target
Leukocyte tyrosine kinase receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LTK kinase domain
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Target
Tyrosine-protein kinase ZAP-70
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ZAP70 kinase domain
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Target Info
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Target
Serine/threonine-protein kinase N1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKN1 kinase domain
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Target
Wee1-like protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for WEE2 kinase domain
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Target
Uncharacterized serine/threonine-protein kinase SBK3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SgK110 kinase domain
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Target
Dual serine/threonine and tyrosine protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RIPK5 kinase domain
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Target
Calcium-dependent protein kinase 1
(Plasmodium Falciparum)
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PFCDPK1(P.falciparum) kinase domain
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Target
Cyclin-dependent kinase 2 homolog
(Plasmodium falciparum (isolate 3D7))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PFPK5(P.falciparum) kinase domain
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Target
Serine/threonine-protein kinase mTOR
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MTOR kinase domain
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Target
Tyrosine-protein kinase JAK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JAK2(JH1domain-catalytic) kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CD kinase domain
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Target
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PLK1 kinase domain
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Target Info
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Target
cAMP-dependent protein kinase catalytic subunit PRKX
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKX kinase domain
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Target Info
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Target
Serine/threonine-protein kinase OSR1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for OSR1 kinase domain
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 2.30E+3nM
Assay Description:
Binding constant for ABL1(F317L)-phosphorylated kinase domain
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Target
Tyrosine-protein kinase ABL2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.80E+3nM
Assay Description:
Binding constant for ABL2 kinase domain
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Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AKT1 kinase domain
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Target
Macrophage colony-stimulating factor 1 receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.90E+3nM
Assay Description:
Binding constant for CSF1R kinase domain
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 5.30E+3nM
Assay Description:
Binding constant for EGFR(L861Q) kinase domain
More data for this Ligand-Target Pair
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Target
Ephrin type-A receptor 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA3 kinase domain
More data for this Ligand-Target Pair
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Target
Tyrosine-protein kinase Fer
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for FER kinase domain
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Target
Tyrosine-protein kinase Fgr
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for FGR kinase domain
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Target
Cyclin-G-associated kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for GAK kinase domain
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 1.10E+3nM
Assay Description:
Binding constant for LCK kinase domain
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Target
Protein kinase C epsilon type
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKCE kinase domain
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Target
Rho-associated protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ROCK1 kinase domain
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Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 1.60E+3nM
Assay Description:
Binding constant for SRC kinase domain
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Target
Tyrosine-protein kinase receptor Tie-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 1.10E+3nM
Assay Description:
Binding constant for TIE1 kinase domain
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Target
Tyrosine-protein kinase Yes
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for YES kinase domain
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Target
RAC-gamma serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AKT3 kinase domain
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Target
Tyrosine-protein kinase ITK/TSK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ITK kinase domain
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Target
LIM domain kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LIMK2 kinase domain
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Target
Muscle, skeletal receptor tyrosine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MUSK kinase domain
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Target
Homeodomain-interacting protein kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for HIPK3 kinase domain
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Target
Serine/threonine-protein kinase D3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKD3 kinase domain
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Target
Serine/threonine-protein kinase MAK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MAK kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP3K1 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ASK1 kinase domain
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Target
Protein-tyrosine kinase 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for BRK kinase domain
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Target
Serine/threonine-protein kinase 10
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 220nM
Assay Description:
Binding constant for LOK kinase domain
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Target
Serine/threonine-protein kinase MRCK beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MRCKB kinase domain
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Target
BDNF/NT-3 growth factors receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TRKB kinase domain
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Target
Cyclin-dependent kinase 16
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PCTK1 kinase domain
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Target
Platelet-derived growth factor receptor alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 11nM
Assay Description:
Binding constant for PDGFRA kinase domain
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Target
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PHKG1 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CA(H1047Y) kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CB kinase domain
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Target
5'-AMP-activated protein kinase catalytic subunit alpha-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AMPK-alpha2 kinase domain
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Target
Protein kinase C delta type
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKCD kinase domain
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Target
Serine/threonine-protein kinase N2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKN2 kinase domain
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Target
Protein kinase C theta type
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKCQ kinase domain
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Target
cGMP-dependent protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKG2 kinase domain
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Target
Serine/threonine-protein kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MST2 kinase domain
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Target
Serine/threonine-protein kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MST1 kinase domain
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Target
Dual specificity testis-specific protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TESK1 kinase domain
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Target
Tyrosine-protein kinase receptor TYRO3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TYRO3 kinase domain
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Target
Serine/threonine-protein kinase VRK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for VRK2 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 12
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DLK kinase domain
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Target
Serine/threonine-protein kinase 25
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for YSK1 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase kinase 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.40E+3nM
Assay Description:
Binding constant for MAP4K5 kinase domain
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NCI pathway
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Mitogen-activated protein kinase kinase kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP3K2 kinase domain
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Target
Serine/threonine-protein kinase PLK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PLK2 kinase domain
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Target
Serine/threonine-protein kinase pim-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIM2 kinase domain
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Target
Citron Rho-interacting kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CIT kinase domain
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Target
Serine/threonine-protein kinase TAO1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TAOK1 kinase domain
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Target
Casein kinase I isoform gamma-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1G1 kinase domain
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Target
Homeodomain-interacting protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for HIPK2 kinase domain
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Target
Fibroblast growth factor receptor 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 600nM
Assay Description:
Binding constant for FGFR4 kinase domain
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Target
Fibroblast growth factor receptor 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 110nM
Assay Description:
Binding constant for FGFR2 kinase domain
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 99nM
Assay Description:
Binding constant for FGFR1 kinase domain
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Target
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIP5K2C kinase domain
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Target
Atypical kinase COQ8B, mitochondrial
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ADCK4 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 19
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 500nM
Assay Description:
Binding constant for YSK4 kinase domain
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Target
Dual specificity mitogen-activated protein kinase kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MEK2 kinase domain
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Target
Serine/threonine-protein kinase 33
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 3.20E+3nM
Assay Description:
Binding constant for STK33 kinase domain
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Target
NUAK family SNF1-like kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SNARK kinase domain
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Target
MAP/microtubule affinity-regulating kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MARK4 kinase domain
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Target
Serine/threonine-protein kinase RIO1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RIOK1 kinase domain
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Target
Testis-specific serine/threonine-protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TSSK1B kinase domain
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Target
Calcium/calmodulin-dependent protein kinase kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMKK1 kinase domain
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Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAPKAPK2 kinase domain
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Target
Serine/threonine-protein kinase Nek9
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK9 kinase domain
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Target
Myosin light chain kinase 2, skeletal/cardiac muscle
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MYLK2 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 9
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MLK1 kinase domain
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Target
Serine/threonine-protein kinase DCLK3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DCAMKL3 kinase domain
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Target
Serine/threonine-protein kinase PknB
(Mycobacterium tuberculosis)
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKNB(M.tuberculosis) kinase domain
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Target
Cyclin-dependent kinase 11B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDC2L1 kinase domain
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Target
Tyrosine-protein kinase Srms
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for SRMS kinase domain
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Target
Serine/threonine-protein kinase 35
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 26nM
Assay Description:
Binding constant for STK35 kinase domain
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Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for DYRK1A kinase domain
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Target
Serine/threonine-protein kinase Nek7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK7 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 20
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ZAK kinase domain
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Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK2 kinase domain
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Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for p38-alpha kinase domain
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Target
Mitogen-activated protein kinase 15
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK8 kinase domain
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Target
Casein kinase I isoform delta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1D kinase domain
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Target
Mitogen-activated protein kinase 9
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JNK2 kinase domain
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Target
Tyrosine-protein kinase FRK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FRK kinase domain
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Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for GSK3B kinase domain
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Target
Tyrosine-protein kinase HCK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 2.70E+3nM
Assay Description:
Binding constant for HCK kinase domain
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Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for JAK1(JH1domain-catalytic) kinase domain
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 5nM
Assay Description:
Binding constant for VEGFR2 kinase domain
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Target
LIM domain kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LIMK1 kinase domain
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Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LYN kinase domain
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Target
Megakaryocyte-associated tyrosine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CTK kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP3K3 kinase domain
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Target
Cyclin-dependent kinase 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK5 kinase domain
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Target
Dual specificity protein kinase CLK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CLK1 kinase domain
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Target
NT-3 growth factor receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TRKC kinase domain
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Target
Mitogen-activated protein kinase 12
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for p38-gamma kinase domain
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Target
Tyrosine-protein kinase Mer
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MERTK kinase domain
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Target
Aurora kinase C
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for AURKC kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type II subunit delta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK2D kinase domain
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Target
Serine/threonine-protein kinase tousled-like 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TLK2 kinase domain
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Target
5'-AMP-activated protein kinase catalytic subunit alpha-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AMPK-alpha1 kinase domain
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Target
Serine/threonine-protein kinase SIK3 [59-1321]
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for QSK kinase domain
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Target
Serine/threonine-protein kinase 16
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for STK16 kinase domain
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Target
Cyclin-dependent kinase 17
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PCTK2 kinase domain
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Target
Discoidin domain-containing receptor 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DDR2 kinase domain
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Target
Serine/threonine-protein kinase receptor R3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ACVRL1 kinase domain
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Target
Tyrosine-protein kinase BTK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for BTK kinase domain
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Target Info
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NCI pathway
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Target
Cyclin-dependent kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK4-cyclinD1 kinase domain
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Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 160nM
Assay Description:
Binding constant for FGFR3 kinase domain
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Target
Tyrosine-protein kinase JAK3
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JAK3(JH1domain-catalytic) kinase domain
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 35nM
Assay Description:
Binding constant for KIT(V559D) kinase domain
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MET(M1250T) kinase domain
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Target
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PHKG2 kinase domain
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Target
Serine/threonine-protein kinase STK11
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for LKB1 kinase domain
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Target Info
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Target
Angiopoietin-1 receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 440nM
Assay Description:
Binding constant for TIE2 kinase domain
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Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for IGF1R kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 15
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP3K15 kinase domain
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Target
Serine/threonine-protein kinase pim-3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PIM3 kinase domain
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Target
Serine/threonine-protein kinase Chk2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CHEK2 kinase domain
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Target
Receptor tyrosine-protein kinase erbB-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERBB2 kinase domain
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Target
Ribosomal protein S6 kinase alpha-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK3(Kin.Dom.1-N-terminal) kinase domain
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Target
Ribosomal protein S6 kinase alpha-4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RPS6KA4(Kin.Dom.2-C-terminal) kinase domain
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Target Info
NCI pathway
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Target
Activated CDC42 kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TNK2 kinase domain
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Target Info
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Target
High affinity nerve growth factor receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TRKA kinase domain
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Target
Myosin light chain kinase family member 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MYLK4 kinase domain
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Target
Serine/threonine-protein kinase PAK 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK4 kinase domain
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Target Info
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Target
Serine/threonine-protein kinase SBK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SBK1 kinase domain
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Target
Serine/threonine-protein kinase DCLK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DCAMKL2 kinase domain
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Target
Receptor tyrosine-protein kinase erbB-4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERBB4 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for HPK1 kinase domain
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Target
Serine/threonine-protein kinase ULK3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ULK3 kinase domain
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Target
Activin receptor type-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ACVR1 kinase domain
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Target
Activin receptor type-2B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ACVR2B kinase domain
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Target
Serine/threonine-protein kinase 32A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for YANK1 kinase domain
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Target
Cyclin-dependent kinase-like 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDKL3 kinase domain
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Target
MAP kinase-interacting serine/threonine-protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MKNK1 kinase domain
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Target
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIP5K1A kinase domain
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Target
Bone morphogenetic protein receptor type-1B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BMPR1B kinase domain
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Target
Bone morphogenetic protein receptor type-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for BMPR2 kinase domain
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Target
Cyclin-dependent kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK3 kinase domain
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Target
Cyclin-dependent kinase 8
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK8 kinase domain
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Target
Cyclin-dependent kinase 9
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK9 kinase domain
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Target
Casein kinase I isoform gamma-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1G2 kinase domain
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Target
Death-associated protein kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DAPK3 kinase domain
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Target
Serine/threonine-protein kinase/endoribonuclease IRE1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERN1 kinase domain
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Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for IKK-beta kinase domain
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Target
Interleukin-1 receptor-associated kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for IRAK1 kinase domain
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Target
Activin receptor type-2A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ACVR2A kinase domain
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Target
RAC-beta serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AKT2 kinase domain
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Target
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AXL kinase domain
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Target
Tyrosine-protein kinase Blk
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 2.00E+3nM
Assay Description:
Binding constant for BLK kinase domain
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Target
Cytoplasmic tyrosine-protein kinase BMX
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BMX kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type IV
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK4 kinase domain
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Target
Cyclin-dependent kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK2 kinase domain
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Target
Cyclin-dependent kinase 7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK7 kinase domain
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Target
Casein kinase I isoform alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1A1 kinase domain
More data for this Ligand-Target Pair
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Target
Casein kinase I isoform epsilon
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1E kinase domain
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Target
Casein kinase II subunit alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK2A1 kinase domain
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Target
Casein kinase II subunit alpha'
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK2A2 kinase domain
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Target
Epithelial discoidin domain-containing receptor 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 160nM
Assay Description:
Binding constant for DDR1 kinase domain
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Target
Receptor tyrosine-protein kinase erbB-3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERBB3 kinase domain
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Target
Tyrosine-protein kinase Fes/Fps
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for FES kinase domain
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 10nM
Assay Description:
Binding constant for FLT1 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MLK3 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 10
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MLK2 kinase domain
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Target
Serine/threonine-protein kinase Nek2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK2 kinase domain
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Target
Serine/threonine-protein kinase Nek3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK3 kinase domain
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Target
Serine/threonine-protein kinase PAK 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK1 kinase domain
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Target
Serine/threonine-protein kinase PAK 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK2 kinase domain
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Target
Serine/threonine-protein kinase PAK 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK3 kinase domain
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Target
Cyclin-dependent kinase 18 [3-474]
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PCTK3 kinase domain
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Target
Platelet-derived growth factor receptor beta
(Homo sapiens (Human))
Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 50nM
Assay Description:
Binding constant for PDGFRB kinase domain
More data for this Ligand-Target Pair
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Target
3-phosphoinositide-dependent protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PDPK1 kinase domain
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Target
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3C2B kinase domain
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Target
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PIM1 kinase domain
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3CG kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Phosphatidylinositol 4-kinase beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK4CB kinase domain
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Target
cAMP-dependent protein kinase catalytic subunit alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKAC-alpha kinase domain
More data for this Ligand-Target Pair
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Target
cAMP-dependent protein kinase catalytic subunit beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PKAC-beta kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Protein kinase C iota type
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKCI kinase domain
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Target
Serine/threonine-protein kinase D1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKD1 kinase domain
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Target Info
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Target
Mitogen-activated protein kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Mitogen-activated protein kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK4 kinase domain
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Target
Mitogen-activated protein kinase 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK3 kinase domain
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Target Info
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Target
Mitogen-activated protein kinase 7
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ERK5 kinase domain
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Target
Mitogen-activated protein kinase 8
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JNK1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Mitogen-activated protein kinase 11
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for p38-beta kinase domain
More data for this Ligand-Target Pair
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Target
Mitogen-activated protein kinase 10
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for JNK3 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Mitogen-activated protein kinase 13
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for p38-delta kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Dual specificity mitogen-activated protein kinase kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MEK1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Dual specificity mitogen-activated protein kinase kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MEK3 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Dual specificity mitogen-activated protein kinase kinase 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MEK6 kinase domain
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Target Info
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Target
Interferon-induced, double-stranded RNA-activated protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PRKR kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
RAF proto-oncogene serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RAF1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Rhodopsin kinase GRK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for GRK1 kinase domain
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Target Info
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Target
Proto-oncogene tyrosine-protein kinase ROS
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ROS1 kinase domain
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Target
Ribosomal protein S6 kinase alpha-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK1(Kin.Dom.1-N-terminal) kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Dual specificity mitogen-activated protein kinase kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MEK4 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
SRSF protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SRPK1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Serine/threonine-protein kinase Nek4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK4 kinase domain
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Target
Cyclin-dependent kinase-like 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDKL5 kinase domain
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Target
Ribosomal protein S6 kinase beta-1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for S6K1 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SYK kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase Tec
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TEC kinase domain
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Target
TGF-beta receptor type-2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TGFBR2 kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Dual specificity protein kinase TTK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TTK kinase domain
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase TXK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TXK kinase domain
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Target
Non-receptor tyrosine-protein kinase TYK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TYK2(JH1domain-catalytic) kinase domain
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Target
Wee1-like protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for WEE1 kinase domain
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Target
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIP5K2B kinase domain
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Target
Serine/threonine-protein kinase ULK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ULK1 kinase domain
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Target
Serine/threonine-protein kinase 24
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MST3 kinase domain
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Target
Dual specificity tyrosine-phosphorylation-regulated kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DYRK2 kinase domain
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Target
Aurora kinase A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for AURKA kinase domain
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Target
Serine/threonine-protein kinase MRCK alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MRCKA kinase domain
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Target
Mitogen-activated protein kinase kinase kinase kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP4K3 kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK1 kinase domain
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Target
MAP kinase-activated protein kinase 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAPKAPK5 kinase domain
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Target
Peripheral plasma membrane protein CASK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CASK kinase domain
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Target
Cyclin-dependent kinase 13
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDC2L5 kinase domain
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Target
Receptor-interacting serine/threonine-protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RIPK1 kinase domain
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Target
Receptor-interacting serine/threonine-protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 2.90E+3nM
Assay Description:
Binding constant for RIPK2 kinase domain
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Target
Serine/threonine-protein kinase RIO3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RIOK3 kinase domain
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Target
Serine/threonine-protein kinase PRP4 homolog
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PRP4 kinase domain
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Target
Cyclin-dependent kinase-like 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDKL2 kinase domain
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Target
Serine/threonine-protein kinase BRSK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BRSK2 kinase domain
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Target
Non-receptor tyrosine-protein kinase TNK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TNK1 kinase domain
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Target
Dual specificity protein kinase CLK3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CLK3 kinase domain
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Target
Dual specificity protein kinase CLK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CLK2 kinase domain
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Target
Serine/threonine-protein kinase PLK3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PLK3 kinase domain
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for FLT3(R834Q) kinase domain
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Target
Cyclin-dependent kinase-like 1 [2-358]
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CDKL1 kinase domain
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Target
Serine/threonine-protein kinase 17B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DRAK2 kinase domain
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Target
Activin receptor type-1B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ACVR1B kinase domain
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Target
ALK tyrosine kinase receptor
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ALK kinase domain
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Target
Bone morphogenetic protein receptor type-1A
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BMPR1A kinase domain
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Target
Serine/threonine-protein kinase B-raf
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for BRAF(V600E) kinase domain
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Target
Tyrosine-protein kinase CSK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CSK kinase domain
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Target
Casein kinase I isoform gamma-3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CSNK1G3 kinase domain
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Target
Ephrin type-A receptor 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA2 kinase domain
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Target Info
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Target
Ephrin type-A receptor 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA4 kinase domain
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Target Info
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Target
Ephrin type-A receptor 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.70E+3nM
Assay Description:
Binding constant for EPHA7 kinase domain
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Target
Ephrin type-B receptor 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHB1 kinase domain
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Target
Ephrin type-B receptor 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHB3 kinase domain
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Target
Ephrin type-B receptor 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHB4 kinase domain
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Target Info
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Target
Ephrin type-B receptor 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 1.40E+3nM
Assay Description:
Binding constant for EPHB6 kinase domain
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Target
Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIK3C2G kinase domain
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Target
Mitogen-activated protein kinase kinase kinase kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MAP4K2 kinase domain
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Target
Ribosomal protein S6 kinase alpha-3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK2(Kin.Dom.1-N-terminal) kinase domain
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Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TGFBR1 kinase domain
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Target Info
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Target
Serine/threonine-protein kinase 38
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NDR1 kinase domain
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Target
Serine/threonine-protein kinase Nek1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK1 kinase domain
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Target
Serine/threonine-protein kinase tousled-like 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TLK1 kinase domain
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Target
Cyclin-dependent kinase 14
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PFTK1 kinase domain
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Target
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PIP5K1C kinase domain
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Target
STE20/SPS1-related proline-alanine-rich protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for STK39 kinase domain
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Target
Serine/threonine-protein kinase TBK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for TBK1 kinase domain
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Target
Serine/threonine-protein kinase Sgk3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for SGK3 kinase domain
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Target Info
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Target
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for IKK-epsilon kinase domain
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Target
Insulin receptor-related protein
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for INSRR kinase domain
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Target
Serine/threonine-protein kinase PLK4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for PLK4 kinase domain
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Target Info
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Target
Death-associated protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for DAPK2 kinase domain
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Target
SRSF protein kinase 3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for SRPK3 kinase domain
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Target
Serine/threonine-protein kinase Nek6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for NEK6 kinase domain
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Target
Eukaryotic translation initiation factor 2-alpha kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for EIF2AK1 kinase domain
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Target
Ribosomal protein S6 kinase alpha-6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RSK4(Kin.Dom.1-N-terminal) kinase domain
More data for this Ligand-Target Pair
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Target
Serine/threonine-protein kinase LATS2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for LATS2 kinase domain
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Target Info
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Target
Hormonally up-regulated neu tumor-associated kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for HUNK kinase domain
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Target
Serine/threonine-protein kinase ULK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ULK2 kinase domain
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Target
STE20-like serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 170nM
Assay Description:
Binding constant for SLK kinase domain
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Target
Maternal embryonic leucine zipper kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for MELK kinase domain
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Target
NUAK family SNF1-like kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for ARK5 kinase domain
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Target
Serine/threonine-protein kinase ICK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ICK kinase domain
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Target
Microtubule-associated serine/threonine-protein kinase 1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MAST1 kinase domain
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Target
Serine/threonine-protein kinase 38-like
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for NDR2 kinase domain
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Target
TRAF2 and NCK-interacting protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 160nM
Assay Description:
Binding constant for TNIK kinase domain
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Target
Cyclin-dependent kinase 19
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CDK11 kinase domain
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Target
Serine/threonine-protein kinase SIK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for SIK2 kinase domain
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Target
Serine/threonine-protein kinase 36
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for STK36 kinase domain
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Target
Interleukin-1 receptor-associated kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for IRAK4 kinase domain
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Target
Serine/threonine-protein kinase TAO2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TAOK2 kinase domain
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Target
Serine/threonine-protein kinase NLK
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for NLK kinase domain
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Target
Serine/threonine-protein kinase TAO3
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TAOK3 kinase domain
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Target
Serine/threonine-protein kinase 26
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MST4 kinase domain
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Target
Myosin-IIIa
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MYO3A kinase domain
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Target
Ephrin type-B receptor 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHB2 kinase domain
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Target
Serine/threonine-protein kinase MARK2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MARK2 kinase domain
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Target
MAP kinase-interacting serine/threonine-protein kinase 2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MKNK2 kinase domain
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Target
BMP-2-inducible protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for BIKE kinase domain
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Target
Transient receptor potential cation channel subfamily M member 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for TRPM6 kinase domain
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Target
SNF-related serine/threonine-protein kinase
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for SNRK kinase domain
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Target
Serine/threonine-protein kinase RIO2
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for RIOK2 kinase domain
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Target
Serine/threonine-protein kinase 32B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: 3.90E+3nM
Assay Description:
Binding constant for YANK2 kinase domain
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Target
Serine/threonine-protein kinase MARK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for MARK1 kinase domain
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Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for GSK3A kinase domain
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Target
Serine/threonine-protein kinase PAK 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK6 kinase domain
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Target
Atypical kinase COQ8A, mitochondrial
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ADCK3 kinase domain
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Target
Serine/threonine-protein kinase PAK 5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for PAK7 kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 6
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for ASK2 kinase domain
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Target
Serine/threonine-protein kinase LATS1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LATS1 kinase domain
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Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for DYRK1B kinase domain
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Target
Mitogen-activated protein kinase kinase kinase 13
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for LZK kinase domain
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Target
Serine/threonine-protein kinase DCLK1
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for DCAMKL1 kinase domain
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Target
Ribosomal protein S6 kinase alpha-5
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for RPS6KA5(Kin.Dom.2-C-terminal) kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type 1D
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK1D kinase domain
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Target
Calcium/calmodulin-dependent protein kinase type 1G
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for CAMK1G kinase domain
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Target
Ephrin type-A receptor 8
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Kd: >1.00E+4nM
Assay Description:
Binding constant for EPHA8 kinase domain
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Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Affinity Data
Kd: 390nM
Assay Description:
Binding constant for RET kinase domain
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
MCE
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Receptor-interacting serine/threonine-protein kinase 4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
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Copy InChI
Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for RIPK4 kinase domain
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
MCE
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dual specificity protein kinase CLK4
(Homo sapiens (Human))
Ambit Biosciences
Curated by
ChEMBL
Ligand
BDBM50184807
((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-me...)
Copy SMILES
Copy InChI
Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding constant for CLK4 kinase domain
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
MCE
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
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