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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
46
hits in this display
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0900nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0900nM
Assay Description:
Inhibition of GSK3alpha (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM50613245
(CHEMBL5266553)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.100nM
Assay Description:
Inhibition of full length GST-tagged human recombinant GSK3-alpha using FL-KRREILSRRP[ps]ERYR-NH2 as substrate incubated for 20 hrs
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.200nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.200nM
Assay Description:
Inhibition of GSK3beta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.300nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM50613246
(CHEMBL5316226)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.340nM
Assay Description:
Inhibition of full length GST-tagged human recombinant GSK3-alpha using FL-KRREILSRRP[ps]ERYR-NH2 as substrate incubated for 20 hrs
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.350nM
Assay Description:
Inhibition of full length GST-tagged human recombinant GSK3-alpha using FL-KRREILSRRP[ps]ERYR-NH2 as substrate incubated for 20 hrs
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Glycogen synthase kinase-3 alpha
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.400nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.75nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.800nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM50613245
(CHEMBL5266553)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.20nM
Assay Description:
Inhibition of tau 4R1N phosphorylation (unknown origin) at S396 residue transfected in human U2OS cells coexpressing GFP-tagged beta catenin incubate...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.20nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.20nM
Assay Description:
Inhibition of Tau (unknown origin) phosphorylation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 58nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 58nM
Assay Description:
Inhibition of tau 4R1N phosphorylation (unknown origin) at S396 residue transfected in human U2OS cells coexpressing GFP-tagged beta catenin incubate...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM50613246
(CHEMBL5316226)
Copy SMILES
Copy InChI
Affinity Data
IC50: 86nM
Assay Description:
Inhibition of tau 4R1N phosphorylation (unknown origin) at S396 residue transfected in human U2OS cells coexpressing GFP-tagged beta catenin incubate...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Microtubule-associated protein tau
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 86nM
Assay Description:
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 200nM
Assay Description:
Inhibition of AAK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Protein kinase C theta type
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 360nM
Assay Description:
Inhibition of PKCtheta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 380nM
Assay Description:
Inhibition of PIM1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Cyclin-dependent kinase 2
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.40E+3nM
Assay Description:
Inhibition of CDK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase JAK2
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of JAK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Non-receptor tyrosine-protein kinase TYK2
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of TYK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase TXK
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of TXK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Nuclear receptor subfamily 4 group A member 3
(Homo sapiens)
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of TEC (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of SYK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of p38alpha (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of LynA (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Interleukin-1 receptor-associated kinase 1
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of IRAK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
Copy BDB DOI
Target
Interleukin-1 receptor-associated kinase 4
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of IRAK4 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
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PubMed
Copy BDB DOI
Target
Aurora kinase B
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of Aurora B (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
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PubMed
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Target
Cytoplasmic tyrosine-protein kinase BMX
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of BMX (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
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PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase BTK
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of BTK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
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PubMed
Copy BDB DOI
Target
Casein kinase II subunit alpha
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Copy SMILES
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of CK2A1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
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PubMed
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Target
Casein kinase II subunit alpha'
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of CK2A2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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DrugBank
antibodypedia
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Ligand Info
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PubMed
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Target
Tyrosine-protein kinase ITK/TSK
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of ITK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of JAK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >2.00E+3nM
Assay Description:
Inhibition of LCK (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
antibodypedia
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Target
Cyclin-dependent kinase 5
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: 6.40E+3nM
Assay Description:
Inhibition of CDK5 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Target
Platelet-derived growth factor receptor beta
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of PDGFRbeta (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of MK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
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antibodypedia
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Target
Aurora kinase A
(Mus musculus (mouse))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of mouse AURA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
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Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of IGF1R (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of cKIT (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Target
Ribosomal protein S6 kinase alpha-1
(Homo sapiens (Human))
TBA
Ligand
BDBM610463
(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of RSK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
PubMed
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