Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 17 hits in this display
IC50: 238nMAssay Description:Inhibition of recombinant His-tagged human FLT3 cytoplasmic domain expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: 383nMAssay Description:Inhibition of recombinant His-tagged human TrkA cytoplasmic domain (441 to 796 residues) expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: 448nMAssay Description:Inhibition of recombinant His-tagged human AXL (473 to end residues) cytoplasmic domain expressed in insect cells by FRET assayMore data for this Ligand-Target Pair
IC50: 665nMAssay Description:Inhibition of recombinant GST-tagged human EphA7 cytoplasmic domain expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: 1.22E+3nMAssay Description:Inhibition of recombinant His-tagged human CSF1R cytoplasmic domain (538 to 910 residues) expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: 5.15E+3nMAssay Description:Inhibition of recombinant human full length GST-tagged MLK2 expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length GST-tagged human JNK3 expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length His-tagged human JNK2 (473 to end residues) expressed in baculovirus expression system at by FRET assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length His-tagged human JNK1alpha1 expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant human full length GST-tagged MLK3 expressed in baculovirus expression system by FRET assayMore data for this Ligand-Target Pair
Kd: 120nMAssay Description:Binding affinity to full length wild type human LZK (M1 to W966 residues) expressed in mammalian cells by KINOMEscan assayMore data for this Ligand-Target Pair
Kd: 5.10nMAssay Description:Binding affinity to full length wild type human DLK (M1 to P859 residues) expressed in mammalian cells by KINOMEscan assayMore data for this Ligand-Target Pair