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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
csnk1d
(Homo sapiens (Human))
Bayer Aktiengesellschaft
US Patent
Ligand
BDBM625232
(N-{4-[7-(cyclopropylmethyl)-5-methyl-4-oxo-3-pheny...)
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Affinity Data
IC50: 4nM
Assay Description:
Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1D, expressed by baculovirus infected insect cells ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Casein kinase I isoform alpha
(Homo sapiens (Human))
Bayer Aktiengesellschaft
US Patent
Ligand
BDBM625232
(N-{4-[7-(cyclopropylmethyl)-5-methyl-4-oxo-3-pheny...)
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Affinity Data
IC50: 5.20nM
Assay Description:
Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Bayer Aktiengesellschaft
US Patent
Ligand
BDBM625232
(N-{4-[7-(cyclopropylmethyl)-5-methyl-4-oxo-3-pheny...)
Copy SMILES
Affinity Data
IC50: >2.00E+4nM
Assay Description:
For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into either a black low volume 384 well microtiter ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI